SCHEMBL5593121

SCHEMBL5593121

O=C(O)c1ccc(-c2cccc(CO)c2)nc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LDHA P00338 2/20 0.64
CYP4F2 P78329 1/20 0.56
CYP4A11 Q02928 1/20 0.56
P4HA1 P13674 2/20 0.54
P4HTM Q9NXG6 1/20 0.54
HPGDS O60760 2/20 0.51
FYN P06241 6/20 0.50
PTGER4 P35408 1/20 0.50
SMN1; SMN2 Q16637 2/20 0.49
TSHR P16473 1/20 0.49
KDM5A P29375 1/20 0.48
KDM2B Q8NHM5 1/20 0.48
KDM4C Q9H3R0 1/20 0.48
KDM5B Q9UGL1 1/20 0.48
ACMSD Q8TDX5 1/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
KDM1A O60341 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL503140 0.86 LDHA (0.79) LDHACYP4F2CYP4A11P4HA1P4HTM
SCHEMBL31243316 0.84 LDHA (0.77) LDHACYP4F2CYP4A11P4HA1P4HTM
SCHEMBL20730171 0.83 FYN (0.48) CYP4F2CYP4A11HPGDSFYNKDM1A
SCHEMBL2540857 0.83 ACMSD (0.51) LDHACYP4F2CYP4A11HPGDSFYN
SCHEMBL5592910 0.81 LDHA (0.67) LDHAP4HA1P4HTMHPGDSSMN1; SMN2
SCHEMBL6562815 0.80 LDHA (0.70) LDHACYP4F2CYP4A11P4HA1P4HTM
SCHEMBL5519447 0.79 KMO (0.63) PTGER4KDM5AKDM2BKDM4CKDM5B
SCHEMBL505455 0.79 LDHA (1.00) LDHAP4HA1P4HTMHPGDSSMN1; SMN2
SCHEMBL2560542 0.79 LDHA (0.68) LDHAP4HA1P4HTMHPGDSFYN
SCHEMBL1543156 0.79 HPGDS (0.76) LDHACYP4F2CYP4A11P4HA1P4HTM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007025775-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO disclosed