SCHEMBL5597474

SCHEMBL5597474

Fc1ccc(N2C[CH]NCC2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.46
TP53 P04637 2/20 0.46
ALDH1A1 P00352 4/20 0.46
MAPT P10636 2/20 0.46
MAPK1 P28482 2/20 0.46
LMNA P02545 1/20 0.46
HTT P42858 1/20 0.46
GFER P55789 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
MAOB P27338 2/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
CASP1 P29466 1/20 0.40
CASP7 P55210 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
POLB P06746 1/20 0.40
HTR1A P08908 2/20 0.39
HTR7 P34969 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13724185 0.81 MAPT (0.47) KDM4ETP53ALDH1A1MAPTMAPK1
SCHEMBL28083181 0.81 ADRB1 (0.60) ALDH1A1LMNAHTTGFERHPGD
SCHEMBL7358977 0.80 HTR3E (0.57) ALDH1A1MAPTMAPK1LMNANPC1
SCHEMBL7354505 0.77 ADRB2 (0.60) ALDH1A1TSHRADRB1
SCHEMBL2107593 0.77 ADRB1 (0.64) ALDH1A1MAPTLMNANPC1RAB9A
SCHEMBL894537 0.75 ADRB1 (0.63) KDM4ETP53ALDH1A1MAPTMAPK1
SCHEMBL233425 0.75 ADRB1 (0.63) KDM4ETP53ALDH1A1MAPTMAPK1
Hydrochloric Acid SCHEMBL714521 0.74 ADRB1 (0.61) KDM4ETP53ALDH1A1MAPTMAPK1
Bromide SCHEMBL10674981 0.74 ADRB1 (0.61) KDM4ETP53ALDH1A1MAPTMAPK1
Hydrochloric Acid SCHEMBL1005870 0.74 ADRB1 (0.61) KDM4ETP53ALDH1A1MAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1982001186-A1 NOVEL BENZOXAZOLINONES,SUBSTITUTED IN THE 6-POSITION BY AN AMINOALCOHOL CHAIN OR AMINO-KETONE CHAIN,THEIR PREPARATION AND THEIR USE IN PHARMACEUTICAL PREPARATIONS BUSCH N 1982-04-15 WO claimed
WO-2018112077-A1 INHIBITORS OF DIHYDROCERAMIDE DESATURASE FOR TREATING DISEASE CENTAURUS THERAPEUTICS (US) 2018-06-21 WO disclosed
EP-1268412-B8 SULPHONAMIDO-SUBSTITUTED BRIDGED BICYCLOALKYL DERIVATIVES MERCK SHARP & DOHME (GB) 2007-02-21 EP disclosed
EP-1268412-A1 SULPHONAMIDO-SUBSTITUTED BRIDGED BICYCLOALKYL DERIVATIVES MERCK SHARP & DOHME LTD. (GB) 2003-01-02 EP disclosed
WO-2001070677-A1 SULPHONAMIDO-SUBSTITUTED BRIDGED BICYCLOALKYL DERIVATIVES MERCK SHARP & DOHME LIMITED (GB) 2001-09-27 WO disclosed