SCHEMBL7358977

SCHEMBL7358977

[CH]1CN(c2ccccc2)CCN1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3E A5X5Y0 1/20 0.57
HTR3B O95264 1/20 0.57
ADRB1 P08588 1/20 0.57
HTR3A P46098 1/20 0.57
HTR3D Q70Z44 1/20 0.57
HTR3C Q8WXA8 1/20 0.57
SIGMAR1 Q99720 1/20 0.57
USP2 O75604 3/20 0.43
CYP2D6 P10635 3/20 0.43
CHRNA7 P36544 2/20 0.42
LMNA P02545 2/20 0.42
HTR1A P08908 1/20 0.42
HTR7 P34969 1/20 0.42
LTA4H P09960 1/20 0.42
TSHR P16473 3/20 0.40
HSD17B10 Q99714 2/20 0.40
ALDH1A1 P00352 2/20 0.40
HTR6 P50406 1/20 0.40
CYP3A4 P08684 2/20 0.39
ALOX15 P16050 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7354505 0.80 ADRB2 (0.60) HTR3EHTR3BADRB1HTR3AHTR3D
SCHEMBL13724185 0.80 MAPT (0.47) HTR3EHTR3BADRB1HTR3AHTR3D
SCHEMBL5597474 0.80 KDM4E (0.46) ADRB1LMNAHTR1AHTR7TSHR
SCHEMBL5539647 0.78 SIGMAR1 (0.45) HTR3EHTR3BADRB1HTR3AHTR3D
SCHEMBL29128246 0.78 HTR3E (0.65) HTR3EHTR3BADRB1HTR3AHTR3D
SCHEMBL28956358 0.78 NPC1 (0.47) LMNAHTR1ALTA4HALDH1A1CYP2C19
SCHEMBL2107593 0.76 ADRB1 (0.64) HTR3EHTR3BADRB1HTR3AHTR3D
Phenylpiperazine SCHEMBL24889 0.73 ADRB1 (1.00) HTR3EHTR3BADRB1HTR3AHTR3D
Phenylpiperazine SCHEMBL55125 0.73 ADRB1 (1.00) HTR3EHTR3BADRB1HTR3AHTR3D
Phenylpiperazine SCHEMBL29135595 0.73 ADRB1 (1.00) HTR3EHTR3BADRB1HTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101541331-A Novel macrolides and ketolides with antimicrobial activity WOCKHARDT RESEARCH CENTER (IN) 2009-09-23 CN claimed
CN-101541331-A Novel macrolides and ketolides with antimicrobial activity WOCKHARDT RESEARCH CENTER (IN) 2009-09-23 CN disclosed
EP-1082308-A1 HETEROCYCLICALLY SUBSTITUTED AMIDES USED AS CALPAIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2001-03-14 EP disclosed
WO-1999054305-A1 HETEROCYCLICALLY SUBSTITUTED AMIDES USED AS CALPAIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1999-10-28 WO disclosed
CN-1046529-A Carbostyril derivative OTSUKA PHARMA CO LTD (JP) 1990-10-31 CN disclosed