SCHEMBL5598221

SCHEMBL5598221

C=CCN1Cc2ccc(C(N)=O)cc2C(CC)C1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAU P00749 1/20 0.38
DRD3 P35462 3/20 0.36
DRD2 P14416 2/20 0.36
HTR1A P08908 1/20 0.34
HTR1D P28221 1/20 0.34
HTR2C P28335 1/20 0.34
OPRM1 P35372 5/20 0.34
OPRD1 P41143 5/20 0.34
OPRK1 P41145 4/20 0.34
MEN1 O00255 1/20 0.34
RAB9A P51151 1/20 0.34
KMT2A Q03164 1/20 0.34
KCNH2 Q12809 1/20 0.34
PTGER4 P35408 1/20 0.34
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
NAMPT P43490 1/20 0.33
HSD17B3 P37058 1/20 0.33
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5598037 0.82 ADRA1D (0.37) DRD3DRD2MEN1RAB9AKMT2A
SCHEMBL7337119 0.78 PLAU (0.67) PLAU
Trifluoroacetic Acid SCHEMBL7338206 0.74 PLAU (0.60) PLAU
SCHEMBL7337131 0.74 PLAU (0.50) PLAUMEN1RAB9AKMT2ANAMPT
SCHEMBL8474346 0.73 PLAU (0.59) PLAUDRD3DRD2HTR1AOPRM1
SCHEMBL8237224 0.72 PLAU (0.48) PLAUMEN1RAB9AKMT2A
SCHEMBL24192442 0.64 CHRNB2 (0.38) MEN1RAB9AKMT2ANAMPT
SCHEMBL22461453 0.64 KRAS (0.42)
SCHEMBL22460911 0.64 CYP1A2 (0.35) OPRK1RAB9AKMT2A
SCHEMBL4200544 0.64 CYP2C9 (0.45) DRD3DRD2OPRM1OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007072041-A1 THERAPEUTIC COMPOUNDS ASTEX THERAPEUTICS LIMITED (GB) 2007-06-28 WO disclosed