SCHEMBL5599702

SCHEMBL5599702

Cc1ccc(C[C@@H]2c3ccccc3C3(CCNCC3)CN2C(=O)C2CCC2)c(C)c1

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 8/20 0.35
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
OPRM1 P35372 1/20 0.31
CYP3A4 P08684 1/20 0.31
LPAR1 Q92633 1/20 0.31
MTNR1B P49286 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5635880 0.81 GRIN2B (0.44) OPRM1
SCHEMBL5780939 0.79 OPRD1 (0.45) OPRM1
SCHEMBL5785483 0.69 SLC6A2 (0.33) SLC6A2SLC6A4OPRM1CYP3A4LPAR1
SCHEMBL5578454 0.68 HDAC1 (0.44)
SCHEMBL5578642 0.67 GRIN2B (0.45)
SCHEMBL5599822 0.66 NOTUM (0.52) HSD11B1
SCHEMBL5599270 0.66 NOTUM (0.33) OPRM1
SCHEMBL5599280 0.64 KCNA3 (0.34) HSD11B1CYP3A4
SCHEMBL5635671 0.63 EED (0.37) OPRM1
SCHEMBL4116754 0.63 ACE (0.35) HSD11B1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005063745-A9 NOVEL SPIROINDOLINE OR SPIROISOQUINOLINE COMPOUNDS, METHODS OF USE AND COMPOSITIONS THEREOF ARENA PHARM INC (US) 2007-02-01 WO claimed