SCHEMBL5599757

SCHEMBL5599757

C=CC[C@H]1N(C(=O)c2ccccc2OC)c2ccccc2C12CCNCC2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.40
ALDH1A1 P00352 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
TP53 P04637 2/20 0.38
THRB P10828 1/20 0.38
LMNA P02545 2/20 0.37
MAPT P10636 1/20 0.37
DRD2 P14416 1/20 0.37
HTT P42858 1/20 0.37
KDM4E B2RXH2 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
MAPK14 Q16539 1/20 0.36
USP2 O75604 1/20 0.35
CYP2D6 P10635 1/20 0.35
TSHR P16473 1/20 0.35
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
HTR1A P08908 1/20 0.35
ADRA1D P25100 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5784794 0.85 RXFP1 (0.42) TP53DRD2CYP2C9CYP2C19MAPK14
SCHEMBL5599482 0.85 HTT (0.37) ALDH1A1SMN1; SMN2LMNAHTTKDM4E
SCHEMBL5599667 0.83 ATM (0.37) SMN1; SMN2DRD2HTTTSHRHTR1A
SCHEMBL5786199 0.81 SIGMAR1 (0.43) SIGMAR1ALDH1A1SMN1; SMN2TP53THRB
SCHEMBL5783958 0.80 PAX8 (0.41) TP53
SCHEMBL5781243 0.79 CYP1A2 (0.36) TP53LMNACYP2C9CYP2C19
SCHEMBL5786887 0.77 GNRHR (0.41) DRD2
SCHEMBL5781865 0.76 BCHE (0.36) ALDH1A1MAPTTSHROPRM1
SCHEMBL5782925 0.76 LMNA (0.39) SIGMAR1ALDH1A1SMN1; SMN2LMNAMAPT
SCHEMBL5778222 0.76 SMYD3 (0.34) SIGMAR1ALDH1A1LMNAMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005063745-A9 NOVEL SPIROINDOLINE OR SPIROISOQUINOLINE COMPOUNDS, METHODS OF USE AND COMPOSITIONS THEREOF ARENA PHARM INC (US) 2007-02-01 WO claimed