SCHEMBL5778222

SCHEMBL5778222

C=CCC1N(C(=O)c2ccccc2F)c2ccc(O)cc2C12CCNCC2

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 2/20 0.34
HTT P42858 2/20 0.32
GNRHR P30968 2/20 0.32
TSHR P16473 2/20 0.31
MAPT P10636 2/20 0.31
ALDH1A1 P00352 1/20 0.31
PAX8 Q06710 1/20 0.31
LMNA P02545 1/20 0.31
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31
OPRM1 P35372 1/20 0.31
OPRD1 P41143 1/20 0.31
OPRK1 P41145 1/20 0.31
PARP1 P09874 1/20 0.31
SIGMAR1 Q99720 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5599482 0.89 HTT (0.37) SMYD3HTTTSHRALDH1A1LMNA
SCHEMBL5783958 0.88 PAX8 (0.41) SMYD3PAX8
SCHEMBL5599317 0.85 GNRHR (0.34) SMYD3HTTGNRHRTSHRPAX8
SCHEMBL5780422 0.84 P2RX7 (0.36) GNRHRALDH1A1KCNH2
SCHEMBL5786885 0.84 GNRHR (0.33) GNRHRKCNH2
SCHEMBL5599667 0.83 ATM (0.37) HTTTSHR
SCHEMBL5786887 0.83 GNRHR (0.41) GNRHRKCNH2
SCHEMBL5781243 0.80 CYP1A2 (0.36) LMNA
SCHEMBL5599502 0.79 GNRHR (0.32) GNRHRKCNH2
SCHEMBL5600190 0.78 GNRHR (0.36) GNRHRLMNAPARP1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1716148-A2 NOVEL SPIROINDOLINE OR SPIROISOQUINOLINE COMPOUNDS, METHODS OF USE AND COMPOSITIONS THEREOF Arena Pharmaceuticals, Inc. (US) 2006-11-02 EP claimed
WO-2005063745-A2 NOVEL SPIROINDOLINE OR SPIROISOQUINOLINE COMPOUNDS, METHODS OF USE AND COMPOSITIONS THEREOF ARENA PHARMACEUTICALS, INC. (US) 2005-07-14 WO claimed