SCHEMBL5608228

SCHEMBL5608228

Nc1cc2c(cc1Cc1ccccc1)N[N]C2=O

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PNP P00491 2/20 0.36
DHFR P00374 1/20 0.36
MPO P05164 3/20 0.36
CYP3A4 P08684 2/20 0.36
TPO P07202 1/20 0.36
EPX P11678 1/20 0.36
PARP1 P09874 1/20 0.36
XDH P47989 1/20 0.35
BCL2 P10415 1/20 0.34
BCL2L1 Q07817 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
ALPL P05186 1/20 0.33
MAOB P27338 1/20 0.33
DAO P14920 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5608564 0.86 MPO (0.39) MPOALDH1A1MAOBDAO
SCHEMBL5608541 0.81 MAPT (0.40) MPOALDH1A1HPGDALPLMAOB
SCHEMBL5608922 0.79 MAOA (0.40) CYP3A4ALDH1A1HPGDMAOB
SCHEMBL5608921 0.75 AR (0.38)
SCHEMBL5618439 0.69 MAPT (0.40) MPOCYP3A4ALDH1A1HPGDALPL
SCHEMBL5608450 0.64 ALDH1A1 (0.39) CYP3A4PARP1ALDH1A1HPGD
SCHEMBL1514183 0.62 HTR2A (0.48) CYP3A4BCL2BCL2L1ALDH1A1MAOB
SCHEMBL6839208 0.62 HTR2A (0.48) CYP3A4BCL2BCL2L1ALDH1A1MAOB
SCHEMBL11495775 0.62 AOC3 (0.43) DHFRMPOCYP3A4TPOEPX
SCHEMBL542553 0.60 HTR2A (0.56) DHFRCYP3A4BCL2BCL2L1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1797042-A1 INDOZOLONE DERIVATIVES AS 11B-HSD1 INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2007-06-20 EP disclosed
WO-2006034804-A1 INDOZOLONE DERIVATIVES AS 11B-HSD1 INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2006-04-06 WO disclosed