SCHEMBL5616636

SCHEMBL5616636

COc1ccc2[nH]cc(CCCCCC(N)=O)c2c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 6/20 0.69
MTNR1B P49286 5/20 0.69
MPO P05164 3/20 0.65
HTR1A P08908 3/20 0.64
CYP2D6 P10635 2/20 0.64
CYP1A2 P05177 2/20 0.64
MAPT P10636 1/20 0.64
TSHR P16473 1/20 0.64
NFKB1 P19838 1/20 0.64
HTR1D P28221 1/20 0.64
HTR1B P28222 1/20 0.64
HTR2A P28223 1/20 0.64
HTR2C P28335 1/20 0.64
HTR7 P34969 1/20 0.64
HTR6 P50406 1/20 0.64
HTR4 Q13639 1/20 0.64
TRPM8 Q7Z2W7 1/20 0.64
BLM P54132 2/20 0.62
PMP22 Q01453 2/20 0.62
NPSR1 Q6W5P4 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16495066 0.95 MTNR1A (0.70) MTNR1AMTNR1BMPOHTR1ACYP2D6
SCHEMBL6952853 0.85 KDM4E (0.71) MTNR1AMTNR1BMPOHTR1ACYP2D6
SCHEMBL8020879 0.85 HTR2A (0.67) MTNR1AMTNR1BMPOHTR1ACYP2D6
SCHEMBL5360884 0.84 CYP2D6 (0.79) MTNR1AMTNR1BMPOHTR1ACYP2D6
SCHEMBL5363947 0.84 CYP2D6 (0.79) MTNR1AMTNR1BMPOHTR1ACYP2D6
SCHEMBL5362738 0.84 CYP2D6 (0.79) MTNR1AMTNR1BMPOHTR1ACYP2D6
SCHEMBL7819940 0.84 HTR1A (0.79) MTNR1AMTNR1BMPOHTR1ACYP2D6
SCHEMBL5368511 0.84 CYP2D6 (0.79) MTNR1AMTNR1BMPOHTR1ACYP2D6
SCHEMBL5350306 0.84 CYP2D6 (0.79) MTNR1AMTNR1BMPOHTR1ACYP2D6
SCHEMBL8717741 0.83 MTNR1A (0.78) MTNR1AMTNR1BMPOHTR1ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007101863-A1 THERAPEUTIC COMBINATION OF A 5HT2 RECEPTOR ANTAGONIST AND OF A 5HT2 RECEPTOR ACTIVATOR MACEF (FR) 2007-09-13 WO disclosed