SCHEMBL5635587

SCHEMBL5635587

O=C(O)N1CCC(c2nnc(Cc3ccccc3)o2)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.52
HTT P42858 1/20 0.52
SMN1; SMN2 Q16637 2/20 0.48
GAA P10253 1/20 0.48
THRB P10828 1/20 0.48
MAPT P10636 3/20 0.47
LMNA P02545 2/20 0.46
TNKS O95271 1/20 0.46
PARP1 P09874 1/20 0.46
PARP2 Q9UGN5 1/20 0.46
CCR5 P51681 1/20 0.43
KCNH2 Q12809 1/20 0.43
ALDH1A1 P00352 3/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
TUBB4A P04350 1/20 0.42
TUBB P07437 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14514081 0.84 SMN1; SMN2 (0.70) TSHRHTTSMN1; SMN2GAATHRB
SCHEMBL315267 0.81 MAPT (0.44) HTTSMN1; SMN2GAATHRBMAPT
SCHEMBL5633461 0.77 HDAC3 (0.62) TSHRMAPTTNKSPARP1PARP2
SCHEMBL16400168 0.77 LMNA (0.40) HTTSMN1; SMN2GAATHRBMAPT
SCHEMBL13543047 0.77 PLAT (0.48) TSHRSMN1; SMN2THRBMAPTTNKS
SCHEMBL315752 0.76 PKM (0.42) HTTSMN1; SMN2GAATHRBMAPT
SCHEMBL314794 0.76 ENPP2 (0.46) HTTSMN1; SMN2GAATHRBMAPT
SCHEMBL2709521 0.76 SMN1; SMN2 (0.55) HTTSMN1; SMN2GAATHRBNPC1
SCHEMBL315417 0.74 ENPP2 (0.48) HTTSMN1; SMN2GAATHRBMAPT
SCHEMBL314745 0.74 L3MBTL1 (0.41) HTTSMN1; SMN2GAATHRBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7217714-B1 CCR5 modulators AGOURON PHARMACEUTICALS, INC. (US) 2007-05-15 US disclosed