SCHEMBL5643285

SCHEMBL5643285

C=C(C(=O)OCC)c1ccc(I)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
MAPT P10636 1/20 0.47
CA1 P00915 4/20 0.42
CA2 P00918 4/20 0.42
CA12 O43570 2/20 0.42
CA7 P43166 2/20 0.42
CA9 Q16790 2/20 0.42
CA14 Q9ULX7 2/20 0.42
KYAT1 Q16773 1/20 0.42
ESR1 P03372 1/20 0.42
ESR2 Q92731 1/20 0.42
TPMT P51580 1/20 0.41
LMNA P02545 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
MAOA P21397 1/20 0.41
TSHR P16473 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
OPRM1 P35372 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5059081 0.91 MAPT (0.55) ALDH1A1MAPTCA1CA2CA12
SCHEMBL5086187 0.85 ALDH1A1 (0.50) ALDH1A1MAPTCA1CA2CA12
SCHEMBL2491603 0.84 CA12 (0.61) ALDH1A1MAPTCA1CA2CA12
SCHEMBL6718454 0.84 ALDH1A1 (0.53) ALDH1A1MAPTCA1CA2CA12
SCHEMBL9141441 0.82 MAPT (0.54) ALDH1A1MAPTCA1CA2CA12
SCHEMBL7079697 0.82 SMN1; SMN2 (0.53) ALDH1A1MAPTLMNACYP1A2CYP3A4
SCHEMBL1966571 0.82 MAPT (0.54) ALDH1A1MAPTCA1CA2CA12
SCHEMBL5626568 0.82 LMNA (0.62) ALDH1A1MAPTCA1CA2CA12
SCHEMBL316956 0.81 ALDH1A1 (0.69) ALDH1A1MAPTLMNATSHRMEN1
SCHEMBL13909369 0.81 ALDH1A1 (0.50) ALDH1A1MAPTCA1CA2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116891461-B Synthesis method of SERD intermediate 罗欣药业(上海)有限公司 2026-05-15 CN disclosed
CN-116891461-A Synthesis method of SERD intermediate 罗欣药业(上海)有限公司 2023-10-17 CN disclosed
CN-108484500-A A kind of preparation method of 1- trifluoroethyls isoquinolin 四川理工学院 2018-09-04 CN disclosed
CN-107400096-A A kind of synthetic method of triazole compounds 湖南华腾制药有限公司 2017-11-28 CN disclosed
CN-106543081-A A kind of preparation method of 1 fluoroalkyl isoquinolin 四川理工学院 2017-03-29 CN disclosed
US-7226951-B2 Compounds having selective cytochrome P450RAI-1 or selective cytochrome P450RAI-2 inhibitory activity and methods of obtaining the same ALLERGAN, INC. (US) 2007-06-05 US disclosed
US-20050176689-A1 Compounds having selective cytochrome P450RAI-1 or selective cytochrome P450RAI-2 inhibitory activity and methods of obtaining the same ALLERGAN, INC. 2005-08-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050176689-A1 Compounds having selective cytochrome P450RAI-1 or selective cytochrome P450RAI-2 inhibitory activity and methods of obtaining the same CYP1A2, CYP2A7, CYP3A7 ALDH1A1 96/4885MAPT 4562/4885CA1 1902/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.