SCHEMBL5666160

SCHEMBL5666160

CCCCOc1ccc(S(=O)(=O)N2CCC3(CC2)[N]C(=O)C(Cc2ccccc2)N3)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.49
L3MBTL1 Q9Y468 2/20 0.49
MAPK1 P28482 2/20 0.49
RECQL P46063 1/20 0.49
ALDH1A1 P00352 3/20 0.41
MMP1 P03956 1/20 0.41
MMP9 P14780 1/20 0.41
MMP13 P45452 1/20 0.41
ADAM17 P78536 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
POLB P06746 1/20 0.40
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
MAPT P10636 1/20 0.40
PKM P14618 1/20 0.40
LMNA P02545 1/20 0.39
HTT P42858 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
TP53 P04637 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5668474 0.89 LMNA (0.52) ALDH1A1KMT2AMEN1PKMLMNA
SCHEMBL5668628 0.87 SMN1; SMN2 (0.41) TSHRL3MBTL1MAPK1ALDH1A1KMT2A
SCHEMBL5668616 0.86 NEK2 (0.49) TSHRL3MBTL1MAPK1ALDH1A1POLB
SCHEMBL5666119 0.82 SMN1; SMN2 (0.39) MAPTPKMLMNAHTTSMN1; SMN2
SCHEMBL4034055 0.80 L3MBTL1 (0.45) TSHRL3MBTL1MAPK1RECQLALDH1A1
SCHEMBL5666460 0.79 ALDH1A1 (0.54) TSHRL3MBTL1MAPK1ALDH1A1KMT2A
SCHEMBL3919279 0.79 L3MBTL1 (0.44) TSHRL3MBTL1MAPK1RECQLALDH1A1
SCHEMBL5668378 0.75 ALDH1A1 (0.57) TSHRL3MBTL1MAPK1ALDH1A1POLB
SCHEMBL4002141 0.74 KMT2A (0.40) L3MBTL1RECQLALDH1A1POLBKMT2A
SCHEMBL5668669 0.74 LMNA (0.59) TSHRL3MBTL1MAPK1ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730144-A1 SUBSTITUTED 1,4,8-TRIAZASPIRO¬4.5|DECAN-2-ONE COMPOUNDS Grünenthal GmbH (DE) 2006-12-13 EP disclosed
WO-2005095398-A1 SUBSTITUTED 1,4,8-TRIAZASPIRO[4.5]DECAN-2-ONE COMPOUNDS Grünenthal GmbH (DE) 2005-10-13 WO disclosed