SCHEMBL5668474

SCHEMBL5668474

COc1ccc(S(=O)(=O)N2CCC3(CC2)[N]C(=O)C(Cc2ccccc2)N3)cc1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.52
ALDH1A1 P00352 6/20 0.50
HSD11B1 P28845 1/20 0.48
PKM P14618 4/20 0.47
NR3C1 P04150 1/20 0.46
NPC1 O15118 1/20 0.46
PKLR P30613 1/20 0.46
RAB9A P51151 1/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
CCR6 P51684 1/20 0.45
CHRM5 P08912 1/20 0.45
KDM4E B2RXH2 1/20 0.45
NPSR1 Q6W5P4 1/20 0.44
HTT P42858 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5668616 0.90 NEK2 (0.49) ALDH1A1MEN1KMT2AHTT
SCHEMBL5666160 0.89 TSHR (0.49) LMNAALDH1A1PKMMEN1KMT2A
SCHEMBL5668628 0.86 SMN1; SMN2 (0.41) LMNAALDH1A1HSD11B1MEN1KMT2A
SCHEMBL5666460 0.82 ALDH1A1 (0.54) LMNAALDH1A1MEN1KMT2ANPSR1
SCHEMBL3915181 0.81 LMNA (0.55) LMNAALDH1A1HSD11B1PKMNR3C1
SCHEMBL5666899 0.80 SMN1; SMN2 (0.51) LMNAALDH1A1RAB9AMEN1KMT2A
SCHEMBL4035567 0.79 LMNA (0.48) LMNAALDH1A1HSD11B1PKMNR3C1
SCHEMBL5668378 0.78 ALDH1A1 (0.57) LMNAALDH1A1PKMNPC1RAB9A
SCHEMBL5666119 0.77 SMN1; SMN2 (0.39) LMNAPKMNPC1HTT
SCHEMBL3917062 0.77 CHRM5 (0.46) LMNAALDH1A1HSD11B1PKMNR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730144-A1 SUBSTITUTED 1,4,8-TRIAZASPIRO¬4.5|DECAN-2-ONE COMPOUNDS Grünenthal GmbH (DE) 2006-12-13 EP disclosed
WO-2005095398-A1 SUBSTITUTED 1,4,8-TRIAZASPIRO[4.5]DECAN-2-ONE COMPOUNDS Grünenthal GmbH (DE) 2005-10-13 WO disclosed