SCHEMBL5667402

SCHEMBL5667402

Clc1ccc2cc(-c3ccccc3)cnc2c1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 4/20 0.73
PDGFRA P16234 4/20 0.73
NR4A2 P43354 1/20 0.50
ESR2 Q92731 1/20 0.50
ADORA3 P0DMS8 1/20 0.49
ADORA1 P30542 1/20 0.49
MAP4K4 O95819 1/20 0.49
AXL P30530 1/20 0.49
CDK8 P49336 1/20 0.49
CYP2A6 P11509 1/20 0.47
MAPK10 P53779 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
BIRC5 O15392 1/20 0.46
PSMB5 P28074 1/20 0.46
CASP3 P42574 1/20 0.46
SENP7 Q9BQF6 1/20 0.46
SENP6 Q9GZR1 1/20 0.46
CNR1 P21554 1/20 0.46
CNR2 P34972 1/20 0.46
NPC1 O15118 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30644240 1.00 PDGFRB (0.73) PDGFRBPDGFRANR4A2ESR2ADORA3
SCHEMBL26613541 0.86 PDGFRB (0.54) PDGFRBPDGFRAADORA3ADORA1MAP4K4
SCHEMBL31060338 0.84 PDGFRB (1.00) PDGFRBPDGFRANR4A2ESR2MAP4K4
SCHEMBL28191718 0.83 ESR2 (0.59) PDGFRBPDGFRAESR2MAP4K4AXL
SCHEMBL29060493 0.80 PDGFRB (0.66) PDGFRBPDGFRAESR2MAP4K4CYP2A6
SCHEMBL29375315 0.80 PDGFRB (0.66) PDGFRBPDGFRAESR2MAP4K4CYP2A6
SCHEMBL708999 0.79 PDGFRB (0.75) PDGFRBPDGFRAMAP4K4AXLCDK8
SCHEMBL20759765 0.79 PSMB5 (0.63) PDGFRBPDGFRAESR2ADORA3ADORA1
SCHEMBL20741503 0.79 TLR9 (0.58) PDGFRBPDGFRAESR2ADORA3AXL
SCHEMBL26560544 0.79 PDGFRB (0.64) PDGFRBPDGFRAESR2MAP4K4CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260083723-A1 THERAPEUTIC AGENT OR PROPHYLACTIC AGENT FOR AMYOTROPHIC LATERAL SCLEROSIS TORAY INDUSTRIES, INC. (JP) 2026-03-26 US disclosed
US-12570639-B2 Tetrahydroquinoline derivative and medicinal use thereof TORAY INDUSTRIES, INC. (JP) 2026-03-10 US disclosed
EP-4545079-A1 THERAPEUTIC AGENT OR PROPHYLACTIC AGENT FOR AMYOTROPHIC LATERAL SCLEROSIS Toray Industries, Inc. (JP) 2025-04-30 EP disclosed
CN-119403554-A Therapeutic or prophylactic agent for amyotrophic lateral sclerosis 东丽株式会社 2025-02-07 CN disclosed
US-20240116903-A1 TETRAHYDROQUINOLINE DERIVATIVE AND MEDICINAL USE THEREOF TORAY INDUSTRIES, INC. (JP) 2024-04-11 US disclosed
WO-2023249105-A1 THERAPEUTIC AGENT OR PREVENTIVE AGENT FOR DRUG-INDUCED MYOCARDIAL DISORDERS 東レ株式会社 2023-12-28 WO disclosed
WO-2023249106-A1 THERAPEUTIC AGENT OR PROPHYLACTIC AGENT FOR AMYOTROPHIC LATERAL SCLEROSIS 東レ株式会社 2023-12-28 WO disclosed
WO-2023249107-A1 THERAPEUTIC AGENT OR PROPHYLACTIC AGENT FOR PERIPHERAL NERVE DISORDER 東レ株式会社 2023-12-28 WO disclosed
CN-117003695-A Preparation method of 2, 3-disubstituted quinoline derivative 广东工业大学 2023-11-07 CN disclosed
EP-4269392-A1 TETRAHYDROQUINOLINE DERIVATIVE AND MEDICINAL USE THEREOF Toray Industries, Inc. (JP) 2023-11-01 EP disclosed
EP-4269392-A1 TETRAHYDROQUINOLINE DERIVATIVE AND MEDICINAL USE THEREOF Toray Industries, Inc. (JP) 2023-11-01 EP disclosed
CN-116648245-A Tetrahydroquinoline derivative and medical application thereof 东丽株式会社 2023-08-25 CN disclosed
WO-2022138888-A1 TETRAHYDROQUINOLINE DERIVATIVE AND MEDICINAL USE THEREOF 東レ株式会社 2022-06-30 WO disclosed
CN-114031552-A Method for synthesizing substituted quinoline derivative from aromatic aldehyde and aromatic amine participated in DMSO 长沙资材科技有限公司 2022-02-11 CN disclosed
US-20060074105-A1 Substituted quinoline and quinazoline inhibitors of quinone reductase 2 SERENEX, INC. (US) 2006-04-06 US disclosed
WO-2006034235-A2 SUBSTITUTED QUINOLINE AND QUINAZOLINE INHIBITORS OF QUINONE REDUCTASE 2 SERENEX, INC. (US) 2006-03-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060074105-A1 Substituted quinoline and quinazoline inhibitors of quinone reductase 2 NQO2, QTRT1, QTRT2 PDGFRB 4772/4885PDGFRA 4728/4885NR4A2 1356/4885
US-20240116903-A1 TETRAHYDROQUINOLINE DERIVATIVE AND MEDICINAL USE THEREOF AIFM2, TXNRD2, NFE2L2 PDGFRB 3381/4885PDGFRA 3877/4885NR4A2 1226/4885
US-20260083723-A1 THERAPEUTIC AGENT OR PROPHYLACTIC AGENT FOR AMYOTROPHIC LATERAL SCLEROSIS AIFM2, GPX1, SOD1 PDGFRB 3258/4885PDGFRA 3519/4885NR4A2 1685/4885
US-12570639-B2 Tetrahydroquinoline derivative and medicinal use thereof AIFM2, GPX1, GPX4 PDGFRB 2960/4885PDGFRA 3340/4885NR4A2 554/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.