SCHEMBL4035567

SCHEMBL4035567

COc1ccc(S(=O)(=O)N2CCC3(CC2)NC(Cc2ccccc2)C(=O)N3CC(=O)O)cc1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.48
PKM P14618 3/20 0.47
MEN1 O00255 4/20 0.47
KMT2A Q03164 4/20 0.47
ALDH1A1 P00352 5/20 0.46
HSD11B1 P28845 1/20 0.46
CHRM5 P08912 1/20 0.46
KDM4E B2RXH2 1/20 0.46
CYP3A4 P08684 2/20 0.44
USP2 O75604 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
NR3C1 P04150 1/20 0.43
GAA P10253 1/20 0.43
MAPT P10636 1/20 0.43
HTT P42858 1/20 0.43
POLB P06746 1/20 0.43
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3927380 0.91 CYP2D6 (0.45) LMNAMEN1KMT2AALDH1A1CYP3A4
SCHEMBL3915181 0.90 LMNA (0.55) LMNAPKMMEN1KMT2AALDH1A1
SCHEMBL4034055 0.90 L3MBTL1 (0.45) LMNAPKMMEN1KMT2AALDH1A1
SCHEMBL4037894 0.89 ALDH1A1 (0.54) LMNAMEN1KMT2AALDH1A1CYP3A4
SCHEMBL4041277 0.88 KMT2A (0.41) LMNAMEN1KMT2AALDH1A1HSD11B1
SCHEMBL4032408 0.84 ALDH1A1 (0.52) LMNAMEN1KMT2AALDH1A1KDM4E
SCHEMBL3917062 0.83 CHRM5 (0.46) LMNAPKMMEN1KMT2AALDH1A1
SCHEMBL4041475 0.83 MMP2 (0.39) LMNAMEN1KMT2AALDH1A1GAA
SCHEMBL2942516 0.83 SMN1; SMN2 (0.48) LMNAMEN1KMT2AALDH1A1KDM4E
SCHEMBL4041453 0.82 MEN1 (0.42) LMNAMEN1KMT2AALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730144-B1 SUBSTITUTED 1,4,8-TRIAZASPIRO¬4.5 DECAN-2-ONE COMPOUNDS GRUENENTHAL GMBH (DE) 2009-06-10 EP claimed