SCHEMBL5680753

SCHEMBL5680753

CCC(C)c1ccc(Oc2ccccc2S(=O)(=O)Cl)cc1C

nearest known ligand 0.63

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 12/20 0.63
HTR2A P28223 4/20 0.38
SLC6A4 P31645 4/20 0.38
KCNH2 Q12809 3/20 0.35
TRPV4 Q9HBA0 1/20 0.34
ALDH1A1 P00352 1/20 0.34
SCN9A Q15858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5683116 0.87 CASP1 (0.59) CASP1HTR2ASLC6A4KCNH2ALDH1A1
SCHEMBL5682849 0.81 CASP1 (0.60) CASP1ALDH1A1
SCHEMBL21970592 0.78 CASP1 (0.52) CASP1HTR2ASLC6A4KCNH2ALDH1A1
SCHEMBL5678964 0.77 CASP1 (0.86) CASP1
SCHEMBL5678951 0.76 CASP1 (0.54) CASP1HTR2ASLC6A4TRPV4SCN9A
SCHEMBL5679392 0.74 CASP1 (0.58) CASP1HTR2ASLC6A4TRPV4ALDH1A1
SCHEMBL6249693 0.72 CASP1 (0.51) CASP1HTR2ASLC6A4TRPV4ALDH1A1
SCHEMBL5682969 0.72 CASP1 (0.55) CASP1HTR2ASLC6A4TRPV4ALDH1A1
SCHEMBL5680993 0.72 CASP1 (0.47) CASP1
SCHEMBL5682872 0.71 GAA (0.53) SLC6A4ALDH1A1SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0932600-B1 SULFONAMIDE SUBSTITUTED ASPARTIC ACID INTERLEUKIN-1BETA CONVERTING ENZYME INHIBITORS WARNER LAMBERT CO (US) 2006-02-08 EP disclosed
US-6083981-A USEFUL FOR TREATMENT OF STROKE, INFLAMMATORY DISEASES, SEPTIC SHOCK, REPERFUSION INJURY, ALZHEIMER'S DISEASE, SHIGELLOSIS WARNER-LAMBERT COMPANY (US) 2000-07-04 US disclosed
US-6054487-A ADMINISTERING AN INTERLEUKIN-ONE BETA CONVERTING ENZYME SUFFICIENT TO INHIBIT PRODUCTION OF GAMMA-INTERFERON BASF AKTIENGESELLSCHAFT (DE) 2000-04-25 US disclosed