SCHEMBL21970592

SCHEMBL21970592

CCC(C)c1ccc(Oc2ccccc2F)cc1C

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 3/20 0.52
HTR2A P28223 5/20 0.42
SLC6A4 P31645 5/20 0.42
PARP10 Q53GL7 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KCNH2 Q12809 3/20 0.38
LPAR1 Q92633 3/20 0.37
LPAR5 Q9H1C0 3/20 0.37
TSHR P16473 1/20 0.36
GCK P35557 1/20 0.36
MMP14 P50281 1/20 0.36
ALDH1A1 P00352 1/20 0.35
ESR1 P03372 1/20 0.35
CARM1 Q86X55 1/20 0.35
PRMT6 Q96LA8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20084781 0.85 CASP1 (0.40) CASP1HTR2ASLC6A4PARP10L3MBTL1
SCHEMBL20085355 0.83 ALDH1A1 (0.40) CASP1HTR2ASLC6A4PARP10L3MBTL1
SCHEMBL5680753 0.78 CASP1 (0.63) CASP1HTR2ASLC6A4KCNH2ALDH1A1
SCHEMBL20084804 0.77 HTR2A (0.55) HTR2ASLC6A4PARP10KCNH2GCK
SCHEMBL6290582 0.74 SLC6A4 (0.40) CASP1HTR2ASLC6A4L3MBTL1KCNH2
SCHEMBL6289858 0.74 SLC6A4 (0.40) CASP1HTR2ASLC6A4L3MBTL1KCNH2
SCHEMBL18928639 0.73 TSHR (0.39) CASP1TSHR
SCHEMBL16792505 0.73 GCK (0.48) HTR2ASLC6A4PARP10L3MBTL1KCNH2
SCHEMBL30764801 0.73 GCK (0.48) HTR2ASLC6A4PARP10L3MBTL1KCNH2
SCHEMBL25962922 0.72 HTR2A (0.49) HTR2ASLC6A4PARP10KCNH2GCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3312172-B1 AMINOPYRAZOLE DERIVATIVES USEFUL AS SRC KINASE INHIBITORS CHUGAI PHARMACEUTICAL CO LTD (JP) 2020-05-06 EP disclosed