SCHEMBL5690164

SCHEMBL5690164

Cc1ccnc(CCc2ccc(OC(=O)N3CCC(Sc4nnnn4CC(=O)O)CC3)cc2)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 2/20 0.35
NOS2 P35228 2/20 0.35
NOS3 P29474 1/20 0.35
NPY2R P49146 1/20 0.34
TLR9 Q9NR96 1/20 0.33
TLR8 Q9NR97 1/20 0.33
TLR7 Q9NYK1 1/20 0.33
GAA P10253 1/20 0.32
GLA P06280 1/20 0.32
MAPT P10636 1/20 0.32
MAPK1 P28482 1/20 0.32
KDM5C P41229 1/20 0.31
KDM2A Q9Y2K7 1/20 0.31
KDM3A Q9Y4C1 1/20 0.31
FFAR1 O14842 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
USP2 O75604 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5687565 0.93 NOS1 (0.35) NOS1NOS2NOS3NPY2RTLR9
SCHEMBL5690392 0.92 FFAR1 (0.35) NOS1NOS2NOS3NPY2RTLR9
SCHEMBL5688818 0.89 NOS3 (0.34) NOS1NOS2NOS3TLR9TLR8
SCHEMBL5931594 0.89 TSHR (0.37) NOS1NOS2NOS3TLR9TLR8
SCHEMBL5687241 0.88 AOC3 (0.36) NPY2RGAAGLAMAPTMAPK1
SCHEMBL5690369 0.85 NOS3 (0.34) NOS1NOS2NOS3NPY2RTLR9
SCHEMBL5687113 0.85 GAA (0.35) NPY2RGAAGLAMAPTMAPK1
SCHEMBL5690600 0.85 KMT2A (0.41) GAAMAPTMAPK1KDM5CKDM2A
SCHEMBL5688221 0.84 NPY2R (0.35) NPY2RGAAMAPK1NPC1RAB9A
SCHEMBL5688785 0.83 NPY2R (0.35) NPY2RTLR9TLR8TLR7GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060160851-A1 Substituted piperidine carbamates NOVO NORDISK A/S (DK) 2006-07-20 US claimed
EP-1636207-A1 SUBSTITUTED PIPERIDINE CARBAMATES FOR USE AS INHIBITORS OF HORMONE SENSITIVE LIPASE NOVO NORDISK A/S (DK) 2006-03-22 EP claimed
WO-2004111032-A1 SUBSTITUTED PIPERIDINE CARBAMATES FOR USE AS INHIBITORS OF HORMONE SENSITIVE LIPASE NOVO NORDISK A/S (DK) 2004-12-23 WO claimed
US-20060160851-A1 Substituted piperidine carbamates NOVO NORDISK A/S (DK) 2006-07-20 US disclosed
EP-1636207-A1 SUBSTITUTED PIPERIDINE CARBAMATES FOR USE AS INHIBITORS OF HORMONE SENSITIVE LIPASE NOVO NORDISK A/S (DK) 2006-03-22 EP disclosed
WO-2004111032-A1 SUBSTITUTED PIPERIDINE CARBAMATES FOR USE AS INHIBITORS OF HORMONE SENSITIVE LIPASE NOVO NORDISK A/S (DK) 2004-12-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060160851-A1 Substituted piperidine carbamates LIPE, PNLIP, LIPC NOS1 646/4885NOS2 797/4885NOS3 444/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.