SCHEMBL570591

SCHEMBL570591

c1cc(CCn2ccnc2)ccn1

nearest known ligand 0.71

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.66
TBXAS1 P24557 4/20 0.61
CYP19A1 P11511 2/20 0.61
KMT2A Q03164 1/20 0.61
HMOX1 P09601 3/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL409741 0.86 HMOX1 (0.72) CYP11B1TBXAS1CYP19A1KMT2AHMOX1
Bromide SCHEMBL29223796 0.85 HMOX1 (0.70) CYP11B1TBXAS1CYP19A1KMT2AHMOX1
Hydrochloric Acid SCHEMBL7527357 0.85 HMOX1 (0.70) CYP11B1TBXAS1CYP19A1KMT2AHMOX1
SCHEMBL10496235 0.83 TBXAS1 (0.56) CYP11B1TBXAS1CYP19A1KMT2AHMOX1
SCHEMBL27460992 0.83 TBXAS1 (0.60) CYP11B1TBXAS1CYP19A1KMT2AHMOX1
SCHEMBL6987156 0.83 CYP19A1 (0.69) CYP11B1TBXAS1CYP19A1KMT2AHMOX1
SCHEMBL6986190 0.83 HMOX1 (0.79) CYP11B1TBXAS1CYP19A1KMT2AHMOX1
SCHEMBL16719036 0.83 CYP19A1 (0.81) CYP11B1TBXAS1CYP19A1KMT2AHMOX1
SCHEMBL10788342 0.83 TBXAS1 (0.65) TBXAS1CYP19A1KMT2AHMOX1
SCHEMBL4316370 0.83 CYP11B1 (0.69) CYP11B1TBXAS1CYP19A1KMT2AHMOX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120196905-A1 SYNTHETIC COMPOUNDS AND METHODS TO DECREASE NICOTINE SELF-ADMINISTRATION HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2012-08-02 US claimed
WO-2012019093-A1 SYNTHETIC COMPOUNDS AND METHODS TO DECREASE NICOTINE SELF-ADMINISTRATION HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2012-02-09 WO claimed
US-8906943-B2 Synthetic compounds and methods to decrease nicotine self-administration HUMAN BIOMOLECULAR RESEARCH INSTITUTE 2014-12-09 US disclosed
US-8906943-B2 Synthetic compounds and methods to decrease nicotine self-administration HUMAN BIOMOLECULAR RESEARCH INSTITUTE 2014-12-09 US disclosed
US-8906943-B2 Synthetic compounds and methods to decrease nicotine self-administration HUMAN BIOMOLECULAR RESEARCH INSTITUTE 2014-12-09 US disclosed
US-20120196905-A1 SYNTHETIC COMPOUNDS AND METHODS TO DECREASE NICOTINE SELF-ADMINISTRATION HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2012-08-02 US disclosed
US-20120196905-A1 SYNTHETIC COMPOUNDS AND METHODS TO DECREASE NICOTINE SELF-ADMINISTRATION HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2012-08-02 US disclosed
US-20120196905-A1 SYNTHETIC COMPOUNDS AND METHODS TO DECREASE NICOTINE SELF-ADMINISTRATION HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2012-08-02 US disclosed
WO-2012019093-A1 SYNTHETIC COMPOUNDS AND METHODS TO DECREASE NICOTINE SELF-ADMINISTRATION HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2012-02-09 WO disclosed
WO-2012019093-A1 SYNTHETIC COMPOUNDS AND METHODS TO DECREASE NICOTINE SELF-ADMINISTRATION HUMAN BIOMOLECULAR RESEARCH INSTITUTE (US) 2012-02-09 WO disclosed
US-4925851-A ANTITUMOR AGENTS; LEUKEMIA SANDOZ PHARMACEUTICALS CORP. (US) 1990-05-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120196905-A1 SYNTHETIC COMPOUNDS AND METHODS TO DECREASE NICOTINE SELF-ADMINISTRATION SLC6A3, NNT, SLC6A2 CYP11B1 1125/4885TBXAS1 3095/4885CYP19A1 4304/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.