SCHEMBL5711059

SCHEMBL5711059

COc1ccccc1C(=O)Nc1cccc(C(O)CN(C)C(=O)c2cnc(N(C)C)nc2-c2ccccc2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 7/20 0.45
KCNK9 Q9NPC2 7/20 0.45
ABL1 P00519 1/20 0.43
EGFR P00533 1/20 0.43
PDGFRB P09619 1/20 0.43
BCR P11274 1/20 0.43
PDGFRA P16234 1/20 0.43
PRKCA P17252 1/20 0.43
BACE1 P56817 1/20 0.42
MAPK1 P28482 2/20 0.42
POLB P06746 4/20 0.41
KMT2A Q03164 1/20 0.41
KDM4E B2RXH2 2/20 0.41
MAPT P10636 3/20 0.40
LMNA P02545 1/20 0.40
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
HTT P42858 1/20 0.39
TP53 P04637 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3944465 0.90 KCNK3 (0.44) KCNK3KCNK9ABL1EGFRPDGFRB
SCHEMBL1386047 0.87 CASR (0.44) KCNK3KCNK9ABL1EGFRPDGFRB
SCHEMBL1386196 0.81 PDK1 (0.43) MAPK1POLBKMT2AKDM4ELMNA
SCHEMBL3944917 0.79 BACE1 (0.41) KCNK3KCNK9ABL1PDGFRBBCR
SCHEMBL3946988 0.78 MEN1 (0.47) KCNK3KCNK9POLBKMT2AKDM4E
SCHEMBL1383618 0.78 ALOX5 (0.47) MAPK1KMT2ALMNAALDH1A1HPGD
SCHEMBL3951861 0.78 GRM4 (0.41) KCNK3KCNK9ABL1BCRBACE1
SCHEMBL3442836 0.77 ALOX5 (0.40) MAPK1POLBKMT2AKDM4EALDH1A1
SCHEMBL3944601 0.75 KCNK3 (0.44) KCNK3ABL1PDGFRBBCRPDGFRA
SCHEMBL3951875 0.75 MAPT (0.42) KCNK3KCNK9ABL1PDGFRBPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1718632-A1 PYRIMIDINE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS Sanofi-Aventis (FR) 2006-11-08 EP disclosed
WO-2005075458-A1 PYRIMIDINE DERIVATIVES AS OREXIN RECEPTORS ANTAGONISTS SANOFI-AVENTIS (FR) 2005-08-18 WO disclosed