SCHEMBL5715434

SCHEMBL5715434

Cc1cccc(CCN2CCN(C(=O)Oc3ccc(Cc4ncccc4C)cc3)CC2)n1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.42
LMNA P02545 1/20 0.42
SMO Q99835 1/20 0.41
THRB P10828 2/20 0.39
GPR4 P46093 1/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
POLB P06746 1/20 0.38
TRPA1 O75762 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
KCNH2 Q12809 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5714511 0.96 SIGMAR1 (0.41) TP53LMNASMOGPR4MAPT
SCHEMBL6102660 0.94 TP53 (0.42) TP53LMNATHRBPOLBTRPA1
SCHEMBL6102545 0.92 KDM4E (0.45) SMOMAPTHTTKDM4EALDH1A1
SCHEMBL5714381 0.90 TP53 (0.52) TP53LMNASMOTHRBKDM4E
SCHEMBL5714838 0.89 TP53 (0.52) TP53LMNATHRBKDM4EALDH1A1
SCHEMBL5714841 0.89 SIGMAR1 (0.43) THRBKCNH2
SCHEMBL5713860 0.89 TP53 (0.42) TP53LMNASMOGPR4POLB
SCHEMBL5714956 0.87 TP53 (0.54) TP53LMNATHRBKDM4EALDH1A1
SCHEMBL5715423 0.86 LMNA (0.40) TP53LMNASMOTHRBMAPT
SCHEMBL6102347 0.85 KCNH2 (0.43) TP53THRBPOLBKDM4ECYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060160820-A1 Substituted piperazine carbamates NOVO NORDISK A/S (DK) 2006-07-20 US claimed
US-20060160820-A1 Substituted piperazine carbamates NOVO NORDISK A/S (DK) 2006-07-20 US disclosed
EP-1636187-A1 SUBSTITUTED PIPERAZINE CARBAMATES FOR USE AS INHIBITORS OF HORMONE SENSITIVE LIPASE NOVO NORDISK A/S (DK) 2006-03-22 EP disclosed
WO-2004111004-A1 SUBSTITUTED PIPERAZINE CARBAMATES FOR USE AS INHIBITORS OF HORMONE SENSITIVE LIPASE NOVO NORDISK A/S (DK) 2004-12-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060160820-A1 Substituted piperazine carbamates LIPE, PNLIP, LPL TP53 2326/4885LMNA 1939/4885SMO 2203/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.