SCHEMBL5723075

SCHEMBL5723075

CC(=O)Nc1ccc(S(=O)(=O)N2C[C@H](S)C[C@H]2C(=O)NNS(=O)(=O)c2ccc(C)cc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GAA P10253 4/20 0.55
KDM4E B2RXH2 1/20 0.55
L3MBTL1 Q9Y468 2/20 0.53
IDO1 P14902 1/20 0.51
NPC1 O15118 1/20 0.51
ALDH1A1 P00352 6/20 0.50
LMNA P02545 2/20 0.50
MEN1 O00255 1/20 0.50
USP2 O75604 1/20 0.50
KMT2A Q03164 1/20 0.50
MAPK1 P28482 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
MAPT P10636 1/20 0.48
MME P08473 1/20 0.48
ACE P12821 1/20 0.48
ECE1 P42892 1/20 0.48
HTT P42858 2/20 0.46
PKM P14618 2/20 0.45
POLB P06746 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5724342 0.92 ALDH1A1 (0.55) GAAL3MBTL1ALDH1A1LMNAMEN1
SCHEMBL5723356 0.88 ALDH1A1 (0.51) GAAL3MBTL1ALDH1A1LMNAMEN1
SCHEMBL5723144 0.88 ECE1 (0.55) GAAL3MBTL1ALDH1A1LMNASMN1; SMN2
SCHEMBL5722907 0.87 GAA (0.53) GAAL3MBTL1ALDH1A1LMNAKMT2A
SCHEMBL5723752 0.87 ALDH1A1 (0.59) L3MBTL1ALDH1A1LMNAKMT2ASMN1; SMN2
SCHEMBL5722993 0.86 MME (0.57) GAAKDM4EL3MBTL1IDO1NPC1
SCHEMBL5722992 0.86 MME (0.57) GAAKDM4EL3MBTL1IDO1NPC1
SCHEMBL5722877 0.85 MMP1 (0.56) ALDH1A1MMEACEECE1
SCHEMBL5723189 0.85 MMP9 (0.54) ALDH1A1SMN1; SMN2MMEACEECE1
SCHEMBL5723026 0.84 ECE1 (0.48) GAAL3MBTL1ALDH1A1LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1317428-B1 PYRROLIDINE-2-CARBOXYLIC ACID HYDRAZIDE DERIVATIVES FOR USE AS METALLOPROTEASE INHIBITORS HOFFMANN LA ROCHE (CH) 2006-04-19 EP disclosed