SCHEMBL5723668

SCHEMBL5723668

CC(=O)SC1CN(c2nc(CNS(=O)(=O)c3ccccc3)cs2)C1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.48
LMNA P02545 4/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
HTT P42858 3/20 0.44
ALDH1A1 P00352 2/20 0.44
STAT3 P40763 1/20 0.44
TSHR P16473 1/20 0.43
KMT2A Q03164 4/20 0.42
MEN1 O00255 3/20 0.42
MAPT P10636 2/20 0.42
HPGD P15428 1/20 0.39
PKM P14618 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5724121 0.84 KDM4E (0.55) KDM4ELMNASMN1; SMN2HTTALDH1A1
SCHEMBL5723960 0.80 KDM4E (0.50) KDM4ELMNASMN1; SMN2HTTALDH1A1
SCHEMBL5724289 0.75 KDM4E (0.45) KDM4ELMNASMN1; SMN2HTTALDH1A1
SCHEMBL5724161 0.71 DNM1L (0.36)
SCHEMBL5826389 0.71 RAB9A (0.34) KDM4ELMNASMN1; SMN2PKM
SCHEMBL6566997 0.70 KMT2A (0.79) KDM4ELMNASMN1; SMN2HTTALDH1A1
SCHEMBL5724296 0.70 KDM4E (0.44) KDM4ELMNASMN1; SMN2HTTALDH1A1
SCHEMBL5724080 0.67 KDM4E (0.47) KDM4ELMNAALDH1A1KMT2AMEN1
SCHEMBL5724065 0.66 KDM4E (0.55) KDM4ELMNAALDH1A1MAPTHPGD
SCHEMBL5724072 0.66 ACKR3 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1340757-B1 1-METHYLCARBAPENEM DERIVATIVES SANKYO CO (JP) 2006-10-11 EP disclosed
US-7001897-B2 1-methylcarbapenem derivatives SANKYO COMPANY, LIMITED (JP) 2006-02-21 US disclosed
US-20040014962-A1 1-Methylcarbapenem derivatives SANKYO COMPANY, LIMITED (JP) 2004-01-22 US disclosed
EP-1340757-A1 1-METHYLCARBAPENEM DERIVATIVES Sankyo Company, Limited (JP) 2003-09-03 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040014962-A1 1-Methylcarbapenem derivatives CD14, CPT1A, ACMSD KDM4E 328/4885LMNA 3159/4885SMN1; SMN2 1508/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.