SCHEMBL5728602

SCHEMBL5728602

CCC(CCc1ccnn1Cc1ccc(OC)cc1)CNS(=O)(=O)c1ccc(Br)cc1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
EGFR P00533 1/20 0.41
ERBB2 P04626 1/20 0.41
GAA P10253 1/20 0.41
KDM4E B2RXH2 1/20 0.39
LMNA P02545 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
IDO1 P14902 1/20 0.38
MMP1 P03956 1/20 0.37
MMP9 P14780 1/20 0.37
MMP13 P45452 1/20 0.37
ADAM17 P78536 1/20 0.37
TSHR P16473 1/20 0.37
HTT P42858 1/20 0.37
USP2 O75604 1/20 0.37
OPRK1 P41145 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3316459 0.74 PSEN1 (0.53) ALDH1A1SMN1; SMN2EGFRERBB2KDM4E
SCHEMBL3314294 0.71 NPBWR1 (0.45) ALDH1A1SMN1; SMN2KDM4E
SCHEMBL29187835 0.70 ALDH1A1 (0.56) ALDH1A1SMN1; SMN2GAALMNAMEN1
SCHEMBL27884291 0.69 NPBWR1 (0.47) ALDH1A1SMN1; SMN2KDM4E
SCHEMBL5732324 0.68 NPBWR1 (0.46) ALDH1A1SMN1; SMN2GAAKDM4ELMNA
SCHEMBL29259796 0.68 ALDH1A1 (0.86) ALDH1A1SMN1; SMN2EGFRERBB2MEN1
SCHEMBL3914871 0.68 ALDH1A1 (0.76) ALDH1A1SMN1; SMN2EGFRERBB2GAA
SCHEMBL3318304 0.67 NPBWR1 (0.50) ALDH1A1SMN1; SMN2KDM4E
SCHEMBL16578700 0.66 MEN1 (0.44) ALDH1A1KDM4ELMNAMEN1KMT2A
SCHEMBL2052679 0.66 NPBWR1 (0.49) ALDH1A1SMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1709003-A1 HETEROCYCLIC SULFONAMIDE INHIBITORS OF BETA AMYLOID PRODUCTION CONTAINING AN AZOLE Wyeth (US) 2006-10-11 EP disclosed
WO-2005073198-A1 HETEROCYCLIC SULFONAMIDE INHIBITORS OF BETA AMYLOID PRODUCTION CONTAINING AN AZOLE WYETH (US) 2005-08-11 WO disclosed