SCHEMBL5732386

SCHEMBL5732386

CC(C)n1ccc2ccc(C(=O)NN3CCC(Cc4ccccc4)CC3)cc21

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAPK11 Q15759 1/20 0.48
MAPK14 Q16539 1/20 0.48
HDAC6 Q9UBN7 2/20 0.47
SLC6A2 P23975 3/20 0.46
SLC6A4 P31645 3/20 0.46
ACHE P22303 1/20 0.44
KCNH2 Q12809 1/20 0.44
HRH3 Q9Y5N1 1/20 0.44
POLB P06746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5377669 0.92 HDAC6 (0.49) HDAC6SLC6A2SLC6A4ACHEKCNH2
SCHEMBL5733936 0.77 HDAC6 (0.52) HDAC6KCNH2HRH3POLB
SCHEMBL7449374 0.77 CCR3 (0.60) SLC6A2SLC6A4
SCHEMBL1063730 0.77 MGLL (0.58) MAPK14KCNH2HRH3
SCHEMBL7076381 0.75 SIGMAR1 (0.48) HDAC6SLC6A2SLC6A4ACHEKCNH2
SCHEMBL5377733 0.73 F2 (0.54) HDAC6SLC6A2SLC6A4ACHEPOLB
SCHEMBL5374680 0.73 ACHE (0.56) MAPK14SLC6A2SLC6A4ACHE
SCHEMBL231079 0.72 MAPK11 (0.55) MAPK11MAPK14HDAC6POLB
SCHEMBL31636989 0.71 MAPK11 (0.56) MAPK11MAPK14HDAC6POLB
SCHEMBL5373096 0.70 GRIN2B (0.53)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1080078-B1 HETEROCYCLIC COMPOUNDS AND METHODS TO TREAT CARDIAC FAILURE AND OTHER DISORDERS SCIOS INC (US) 2006-02-01 EP disclosed