SCHEMBL5739261

SCHEMBL5739261

CC1(C)C(=O)C(C)(C)c2cc(CCCN3CCN(c4onc5ccccc45)CC3)ccc21

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 7/20 0.40
HTR1D P28221 2/20 0.40
HTR1B P28222 2/20 0.40
PARP1 P09874 4/20 0.38
SIGMAR1 Q99720 2/20 0.38
DRD2 P14416 3/20 0.38
HTR2C P28335 4/20 0.37
HTR2A P28223 2/20 0.37
HTR2B P41595 1/20 0.37
HTR7 P34969 3/20 0.36
DRD4 P21917 1/20 0.36
SLC6A4 P31645 1/20 0.36
DRD3 P35462 1/20 0.36
MMP2 P08253 1/20 0.36
MMP9 P14780 1/20 0.36
MMP13 P45452 1/20 0.36
ADAM17 P78536 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5740933 0.95 HTR2A (0.38) HTR1AHTR1DHTR1BPARP1SIGMAR1
SCHEMBL5738682 0.84 SIGMAR1 (0.38) HTR1AHTR1DHTR1BSIGMAR1DRD2
SCHEMBL6399207 0.84 HTR2A (0.50) HTR1ASIGMAR1DRD2HTR2AHTR7
SCHEMBL5738711 0.80 MEN1 (0.39) HTR1A
SCHEMBL6401030 0.79 HTR7 (0.52) DRD2HTR2AHTR7DRD4
SCHEMBL6401515 0.78 HTR1A (0.56) HTR1ADRD2HTR2AHTR7
SCHEMBL5784362 0.78 HTR1A (0.31) HTR1ADRD2HTR2A
SCHEMBL5738767 0.78 HTR2A (0.51) HTR1ADRD2HTR2A
SCHEMBL5750335 0.78 HTR1A (0.39) HTR1AHTR1DHTR1BDRD2HTR2C
SCHEMBL5738687 0.75 HTR1A (0.41) HTR1AHTR1DHTR1BDRD2HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1697334-A1 HETEROCYCLIC SUBSTITUTED INDANE DERIVATIVES AND RELATED COMPOUNDS FOR THE TREATMENT OF SCHIZOPHRENIA Warner-Lambert Company LLC (US) 2006-09-06 EP disclosed
WO-2005056540-A1 HETEROCYCLIC SUBSTITUTED INDANE DERIVATIVES AND RELATED COMPOUNDS FOR THE TREATMENT OF SCHIZOPHRENIA WARNER-LAMBERT COMPANY LLC (US) 2005-06-23 WO disclosed