SCHEMBL5740488

SCHEMBL5740488

COc1ccccc1-c1cc(Nc2ccc3nc(C)cc(N)c3c2)nc(N)n1

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 2/20 0.57
DOT1L Q8TEK3 4/20 0.55
TERT O14746 5/20 0.54
AGPAT2 O15120 3/20 0.52
OPRL1 P41146 1/20 0.48
HSP90AB1 P08238 1/20 0.47
SYK P43405 1/20 0.46
CYP1A2 P05177 1/20 0.45
CYP2D6 P10635 1/20 0.45
RAB9A P51151 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5741860 0.89 MAPT (0.52) HSP90AA1AGPAT2HSP90AB1CYP1A2CYP2D6
SCHEMBL5740482 0.85 ALOX15 (0.48) HSP90AA1AGPAT2HSP90AB1CYP1A2CYP2D6
SCHEMBL5742562 0.85 MAPT (0.53) HSP90AA1AGPAT2HSP90AB1RAB9A
SCHEMBL5741412 0.85 DOT1L (0.57) DOT1LTERTAGPAT2OPRL1CYP1A2
SCHEMBL5740342 0.85 AGPAT2 (0.59) HSP90AA1AGPAT2HSP90AB1
SCHEMBL5744362 0.84 AGPAT2 (0.46) HSP90AA1AGPAT2HSP90AB1
SCHEMBL5741832 0.83 AGPAT2 (0.46) HSP90AA1AGPAT2HSP90AB1CYP1A2CYP2D6
SCHEMBL5743121 0.83 AGPAT2 (0.55) HSP90AA1AGPAT2HSP90AB1
SCHEMBL5741580 0.82 ACP1 (0.48) HSP90AA1AGPAT2HSP90AB1CYP1A2CYP2D6
SCHEMBL5741949 0.81 TP53 (0.49) HSP90AA1AGPAT2HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339706-B1 N-TYPE CALCIUM CHANNEL ANTAGONISTS FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2006-04-19 EP disclosed