SCHEMBL5744362

SCHEMBL5744362

CCCCCc1cc(N)c2cc(Nc3cc(-c4ccccc4OC)nc(N)n3)ccc2n1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AGPAT2 O15120 5/20 0.46
MCHR1 Q99705 7/20 0.44
HSP90AA1 P07900 2/20 0.43
HSP90AB1 P08238 1/20 0.42
PDPK1 O15530 1/20 0.41
ADORA3 P0DMS8 2/20 0.41
ADORA1 P30542 2/20 0.41
TLR8 Q9NR97 1/20 0.39
CHRNA7 P36544 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5740488 0.84 HSP90AA1 (0.57) AGPAT2HSP90AA1HSP90AB1
SCHEMBL5741860 0.83 MAPT (0.52) AGPAT2HSP90AA1HSP90AB1
SCHEMBL5742562 0.80 MAPT (0.53) AGPAT2HSP90AA1HSP90AB1
SCHEMBL5740482 0.80 ALOX15 (0.48) AGPAT2HSP90AA1HSP90AB1
SCHEMBL5741907 0.79 MCHR1 (0.44) AGPAT2MCHR1PDPK1TLR8
SCHEMBL5740342 0.79 AGPAT2 (0.59) AGPAT2HSP90AA1HSP90AB1
SCHEMBL5741832 0.78 AGPAT2 (0.46) AGPAT2HSP90AA1HSP90AB1PDPK1
SCHEMBL5743121 0.78 AGPAT2 (0.55) AGPAT2HSP90AA1HSP90AB1
SCHEMBL5743256 0.78 MCHR1 (0.59) AGPAT2MCHR1TLR8
SCHEMBL5741580 0.77 ACP1 (0.48) AGPAT2MCHR1HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339706-B1 N-TYPE CALCIUM CHANNEL ANTAGONISTS FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2006-04-19 EP disclosed