SCHEMBL5740595

SCHEMBL5740595

N/N=C1\C(=O)Nc2cccc(Cl)c21

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CES1 P23141 2/20 0.61
TGM2 P21980 10/20 0.48
GALR3 O60755 2/20 0.47
PBRM1 Q86U86 4/20 0.43
IDO1 P14902 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9835981 1.00 CES1 (0.61) CES1TGM2GALR3PBRM1IDO1
SCHEMBL5741222 0.81 POLB (0.51) CES1PBRM1IDO1
SCHEMBL5752424 0.79 CES1 (0.61) CES1TGM2GALR3IDO1
SCHEMBL282066 0.76 CES1 (1.00) CES1TGM2PBRM1
SCHEMBL30716604 0.76 CES1 (1.00) CES1TGM2PBRM1
SCHEMBL5740135 0.75 CES1 (0.58) CES1TGM2
Nitrogen SCHEMBL29242307 0.73 CES1 (0.92) CES1TGM2PBRM1
SCHEMBL11530748 0.72 CES1 (0.61) CES1TGM2GALR3IDO1
SCHEMBL5988948 0.72 CES1 (0.61) CES1TGM2GALR3IDO1
SCHEMBL5989290 0.72 LRRK2 (0.50) GALR3IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1644362-A2 INDOLINONE HYDRAZIDES AS C-MET INHIBITORS Sugen, Inc. (US) 2006-04-12 EP disclosed
US-20060009493-A1 Indolinone hydrazides as c-Met inhibitors SUGEN, INC. 2006-01-12 US disclosed
WO-2005005378-A2 INDOLINONE HYDRAZIDES AS C-MET INHIBITORS SUGEN, INC. (US) 2005-01-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060009493-A1 Indolinone hydrazides as c-Met inhibitors MET, IGF1R, ROS1 CES1 1061/4885TGM2 2673/4885GALR3 982/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.