SCHEMBL5740661

SCHEMBL5740661

Cc1nsc2nc(CCCNCCCNC(=O)OC(C)(C)C)n(Cc3ccccc3)c(=O)c12

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 7/20 0.43
KIF11 P52732 3/20 0.41
KIF23 Q02241 1/20 0.41
GNRHR P30968 1/20 0.40
SIGMAR1 Q99720 2/20 0.39
NPSR1 Q6W5P4 1/20 0.38
BRD4 O60885 1/20 0.37
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
CYP3A4 P08684 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5742421 0.90 KIF11 (0.40) TLR7KIF11KIF23GNRHRBRD4
SCHEMBL5248653 0.88 KIF11 (0.42) TLR7KIF11KIF23GNRHRSIGMAR1
SCHEMBL5246236 0.85 KIF11 (0.52) TLR7KIF11KIF23GNRHRSIGMAR1
SCHEMBL5740939 0.84 KIF11 (0.47) TLR7KIF11KIF23GNRHRSIGMAR1
SCHEMBL5246052 0.83 TLR7 (0.43) TLR7KIF11GNRHRSIGMAR1NPSR1
SCHEMBL3871323 0.82 KIF11 (0.49) TLR7KIF11KIF23SIGMAR1NPSR1
SCHEMBL3863849 0.82 KIF11 (0.49) TLR7KIF11KIF23GNRHRSIGMAR1
SCHEMBL6207102 0.82 KIF11 (0.45) KIF11KIF23NPSR1PDE4APDE4B
SCHEMBL5740657 0.81 KIF11 (0.46) TLR7KIF11KIF23SIGMAR1BRD4
SCHEMBL5248649 0.80 KIF11 (0.45) TLR7KIF11KIF23GNRHRSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1628981-A2 BICYCLICPYRIMIDONES AND THEIR USE TO TREAT DISEASES Bristol-Myers Squibb Company (US) 2006-03-01 EP disclosed
WO-2004106492-A2 BICYCLICPYRIMIDONES AND THEIR USE TO TREAT DISEASES BRISTOL-MYERS SQUIBB COMPANY (US) 2004-12-09 WO disclosed