SCHEMBL5741125

SCHEMBL5741125

Cc1cc2c(s1)CCNC2C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
PNMT P11086 1/20 0.39
MAPKAPK2 P49137 9/20 0.38
MAPKAPK5 Q8IW41 1/20 0.38
GRIA2 P42262 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1011216 0.75 PNMT (0.44) TSHRPNMT
SCHEMBL9207161 0.72 TSHR (0.53) TSHRNPSR1MAPKAPK2GRIA2
Hydrochloric Acid SCHEMBL10489402 0.71 TSHR (0.55) TSHRNPSR1MAPKAPK2GRIA2
SCHEMBL19642816 0.70 SIRT1 (0.41) TSHR
SCHEMBL19643822 0.70 SIRT1 (0.41) TSHR
SCHEMBL25373658 0.69 TSHR (0.60) TSHRNPSR1
SCHEMBL30561807 0.69 TSHR (0.60) TSHRNPSR1
SCHEMBL28143019 0.67 DRD2 (0.59) TSHRNPSR1
SCHEMBL9210495 0.67 PNMT (0.37) TSHRPNMT
SCHEMBL12192723 0.66 MAOA (0.50) TSHRNPSR1MAPKAPK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1723148-A2 THIENO-IMINO ACID DERIVATIVES FOR USE AS MATRIX METALLOPROTEINASE INHIBITORS Sanofi-Aventis Deutschland GmbH (DE) 2006-11-22 EP disclosed
WO-2005073236-A2 THIENO-IMINO ACID DERIVATIVES FOR USE AS MATRIX METALLOPROTEINASE INHIBITORS SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2005-08-11 WO disclosed