SCHEMBL574274

SCHEMBL574274

COc1cc(N(C(=O)OC(C)(C)C)C2CCNCC2)c(C)cc1N

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EHMT2 Q96KQ7 1/20 0.39
HTR4 Q13639 5/20 0.38
QPCT Q16769 1/20 0.33
SLC6A4 P31645 7/20 0.33
SLC6A2 P23975 6/20 0.33
ACHE P22303 2/20 0.33
AAK1 Q2M2I8 3/20 0.32
TACR1 P25103 1/20 0.31
HTR3A P46098 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
PLAT P00750 1/20 0.31
SLC6A3 Q01959 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL574202 0.84 LMNA (0.36) EHMT2MEN1KMT2A
SCHEMBL573598 0.81 QPCT (0.41) EHMT2HTR4QPCTSLC6A4SLC6A2
SCHEMBL4439262 0.80 EPHX2 (0.39) HTR4SLC6A4SLC6A2TACR1MEN1
SCHEMBL4442462 0.80 MEN1 (0.36) SLC6A4SLC6A2TACR1MEN1KMT2A
SCHEMBL4439470 0.80 MEN1 (0.36) SLC6A4SLC6A2TACR1MEN1KMT2A
SCHEMBL5214565 0.78 SLC6A2 (0.37) SLC6A4SLC6A2MEN1KMT2ASLC6A3
SCHEMBL4444981 0.76 SLC6A4 (0.40) SLC6A4SLC6A2TACR1MEN1KMT2A
SCHEMBL4437622 0.76 GAA (0.35) SLC6A4SLC6A2TACR1MEN1KMT2A
SCHEMBL4434907 0.76 TACR1 (0.40) SLC6A4SLC6A2TACR1SLC6A3
SCHEMBL27808000 0.72 TACR1 (0.40) SLC6A4SLC6A2TACR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2601186-A2 4-(1H-INDOL-3-YL)-PYRIMIDINES AS ALK INHIBITORS AstraZeneca AB (SE) 2013-06-12 EP disclosed
WO-2012017239-A2 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2012-02-09 WO disclosed