SCHEMBL5742909

SCHEMBL5742909

CC(C)(CC(O)(Cc1ccccc1)C(=O)Nc1cc(Cl)cc(Cl)c1)c1cc(F)ccc1O

nearest known ligand 0.66

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 19/20 0.66
PGR P06401 17/20 0.66
NR3C2 P08235 10/20 0.66
AR P10275 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4617201 0.91 NR3C1 (0.71) NR3C1PGRNR3C2AR
SCHEMBL5742025 0.90 NR3C1 (0.68) NR3C1PGRNR3C2AR
SCHEMBL5744371 0.90 NR3C1 (0.68) NR3C1PGRNR3C2AR
SCHEMBL5742371 0.88 NR3C1 (0.67) NR3C1PGRNR3C2
SCHEMBL5740910 0.87 NR3C1 (0.65) NR3C1PGRNR3C2AR
SCHEMBL3657148 0.82 NR3C1 (0.59) NR3C1PGRNR3C2
SCHEMBL5740674 0.81 PGR (0.64) NR3C1PGRNR3C2AR
SCHEMBL290544 0.81 NR3C1 (0.62) NR3C1PGRNR3C2AR
SCHEMBL5744672 0.80 NR3C1 (0.67) NR3C1PGRNR3C2AR
SCHEMBL292961 0.80 PGR (1.00) NR3C1PGRNR3C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1467982-B1 GLUCOCORTICOID MIMETICS, METHODS OF MAKING THEM, PHARMACEUTICAL FORMULATIONS CONTAINING THEM, AND USES THEREOF BOEHRINGER INGELHEIM PHARMA (US) 2006-11-22 EP claimed
US-7189758-B2 Glucocorticoid mimetics, methods of making them, pharmaceutical formulations, and uses thereof BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2007-03-13 US disclosed
US-7189758-B2 Glucocorticoid mimetics, methods of making them, pharmaceutical formulations, and uses thereof BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2007-03-13 US disclosed
US-6960581-B2 Glucocorticoid mimetics, methods of making them, pharmaceutical formulations, and uses thereof BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2005-11-01 US disclosed