SCHEMBL5746475

SCHEMBL5746475

NC(=O)c1cccnc1-c1nc2ccc([N+](=O)[O-])cc2s1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ILK Q13418 1/20 0.51
ALDH1A1 P00352 5/20 0.50
CYP3A4 P08684 1/20 0.50
TSHR P16473 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
SMN1; SMN2 Q16637 4/20 0.47
HTT P42858 1/20 0.47
CCNE1 P24864 1/20 0.47
CDK2 P24941 1/20 0.47
CDK5 Q00535 1/20 0.47
CDK5R1 Q15078 1/20 0.47
MAPT P10636 5/20 0.47
NPC1 O15118 3/20 0.47
RAB9A P51151 3/20 0.47
KMT2A Q03164 3/20 0.47
MEN1 O00255 2/20 0.47
KCNH2 Q12809 1/20 0.47
DYRK1A Q13627 1/20 0.46
CA2 P00918 1/20 0.46
CA5A P35218 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5177282 0.83 ILK (0.57) ILKALDH1A1CYP3A4TSHRTDP1
SCHEMBL22130264 0.78 SMN1; SMN2 (0.62) ILKALDH1A1CYP3A4TSHRTDP1
SCHEMBL22130227 0.75 ACP1 (0.44) ILKALDH1A1CYP3A4TSHRTDP1
SCHEMBL2379405 0.74 ALDH1A1 (0.64) ILKALDH1A1CYP3A4TSHRTDP1
SCHEMBL25277063 0.74 MAPT (0.51) ALDH1A1TSHRTDP1SMN1; SMN2MAPT
SCHEMBL30014995 0.74 ILK (0.49) ILKALDH1A1CYP3A4TSHRTDP1
SCHEMBL27993567 0.73 KMT2A (0.60) ALDH1A1TSHRTDP1MAPTNPC1
Hydrochloric Acid SCHEMBL28411118 0.73 MAPT (0.51) ALDH1A1TSHRTDP1SMN1; SMN2HTT
SCHEMBL11784834 0.72 RAB9A (0.58) ILKALDH1A1CYP3A4TSHRTDP1
SCHEMBL2136576 0.72 APP (0.69) ILKALDH1A1CYP3A4TSHRTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020130214-A1 NOVEL HYDRAZONE DERIVATIVE WITH ARYL OR HETEROARYL GROUP SUBSTITUTED AT TERMINAL AMINE GROUP THEREOF AND USE THEREOF 한국과학기술연구원 2020-06-25 WO disclosed
EP-1674466-A1 2,5- and 2,6-disubstituted benzazole analogues useful as protein kinase inhibitors 4SC AG (DE) 2006-06-28 EP disclosed