SCHEMBL5177282

SCHEMBL5177282

NC(=O)c1ccccc1-c1nc2ccc([N+](=O)[O-])cc2s1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ILK Q13418 1/20 0.57
ALDH1A1 P00352 6/20 0.53
CYP3A4 P08684 2/20 0.53
TSHR P16473 2/20 0.53
TDP1 Q9NUW8 1/20 0.53
SMN1; SMN2 Q16637 6/20 0.50
HTT P42858 2/20 0.50
CCNE1 P24864 1/20 0.49
CDK2 P24941 1/20 0.49
CDK5 Q00535 1/20 0.49
CDK5R1 Q15078 1/20 0.49
DYRK1A Q13627 1/20 0.49
CA2 P00918 1/20 0.49
CA5A P35218 1/20 0.49
PDK1 Q15118 1/20 0.49
APP P05067 1/20 0.48
MMP2 P08253 1/20 0.48
MMP9 P14780 1/20 0.48
MMP8 P22894 1/20 0.48
MMP13 P45452 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5768391 0.84 MAPT (0.57) ILKALDH1A1TDP1SMN1; SMN2CA2
SCHEMBL5746475 0.83 ILK (0.51) ILKALDH1A1CYP3A4TSHRTDP1
SCHEMBL29787 0.81 MAPT (0.52) HTTDYRK1ACA2CA5AAPP
SCHEMBL5027039 0.79 MAPT (0.63) ILKALDH1A1TSHRTDP1SMN1; SMN2
SCHEMBL11011564 0.77 MMP13 (0.59) ILKALDH1A1CYP3A4SMN1; SMN2HTT
SCHEMBL30810246 0.77 EPHX2 (0.50) ILKSMN1; SMN2DYRK1AMAPTLMNA
SCHEMBL2136576 0.77 APP (0.69) ILKALDH1A1CYP3A4TSHRTDP1
SCHEMBL2379405 0.77 ALDH1A1 (0.64) ILKALDH1A1CYP3A4TSHRTDP1
Hydrochloric Acid SCHEMBL30810214 0.76 EPHX2 (0.49) ILKSMN1; SMN2DYRK1AMAPTLMNA
SCHEMBL1996999 0.74 APP (0.73) ILKALDH1A1CYP3A4TSHRTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020130214-A1 NOVEL HYDRAZONE DERIVATIVE WITH ARYL OR HETEROARYL GROUP SUBSTITUTED AT TERMINAL AMINE GROUP THEREOF AND USE THEREOF 한국과학기술연구원 2020-06-25 WO disclosed
EP-1833823-A1 2,5- AND 2,6-DISUBSTITUTED BENZAZOLE ANALOGUES USEFUL AS PROTEIN KINASE INHIBITORS 4SC AG (DE) 2007-09-19 EP disclosed
WO-2006069740-A1 2, 5 AND 2, 6-DISUBSTITUTED BENZAZOLE ANALOGUES USEFUL AS PROTEIN KINASE INHIBITORS 4SC AG (DE) 2006-07-06 WO disclosed