SCHEMBL5750896

SCHEMBL5750896

COCCOCOc1ccc(/C=C/C=O)cc1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 2/20 0.41
MAPT P10636 2/20 0.41
PTPN1 P18031 2/20 0.40
TRPA1 O75762 2/20 0.39
CTNNB1 P35222 1/20 0.39
LMNA P02545 1/20 0.39
ALOX5 P09917 1/20 0.39
MAPK1 P28482 1/20 0.39
XDH P47989 1/20 0.39
MTNR1A P48039 1/20 0.38
RECQL P46063 1/20 0.38
AHR P35869 1/20 0.38
APP P05067 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18586638 0.89 PTPN1 (0.46) ALDH1A1KDM4EMAPTPTPN1TRPA1
SCHEMBL2832894 0.89 AHR (0.41) PTPN1CTNNB1AHRAPP
SCHEMBL18586639 0.89 PTPN1 (0.46) ALDH1A1KDM4EMAPTPTPN1TRPA1
SCHEMBL25218117 0.87 ALDH1A1 (0.46) ALDH1A1KDM4EMAPTPTPN1TRPA1
SCHEMBL1524953 0.83 ALDH1A1 (0.52) ALDH1A1KDM4EMAPTCTNNB1LMNA
SCHEMBL9035379 0.80 TRPA1 (0.60) ALDH1A1KDM4EMAPTTRPA1LMNA
SCHEMBL9035381 0.80 TRPA1 (0.60) ALDH1A1KDM4EMAPTTRPA1LMNA
SCHEMBL10477124 0.79 FDPS (0.49) CTNNB1APP
SCHEMBL5750014 0.79 THRB (0.59) ALDH1A1KDM4EMAPT
SCHEMBL7663462 0.79 THRB (0.59) ALDH1A1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1387841-B1 NOVEL AZOLE OR TRIAZOLE DERIVATIVES, METHOD FOR PREPARING THE SAME AND USE THEREOF AS FUNGICIDES AVENTIS PHARMA SA (FR) 2006-03-08 EP disclosed
US-6946460-B2 Azole or triazole derivatives, method for preparing same and use thereof as fungicides AVENTIS PHARMA S.A. (FR) 2005-09-20 US disclosed
US-20050043540-A1 Novel azole or triazole derivatives, method for preparing same and use thereof as fungicides AVENTIS PHARMA S. A, (FR) 2005-02-24 US disclosed
US-20030187267-A1 Novel 1,2,3,4-tetrahydroisoquinoline, their preparation method and their use as fungicides AVENTIS PHARMA S.A. (FR) 2003-10-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050043540-A1 Novel azole or triazole derivatives, method for preparing same and use thereof as fungicides CYP1A2, CYP1B1, CYP21A2 ALDH1A1 410/4885KDM4E 2311/4885MAPT 3283/4885
US-20030187267-A1 Novel 1,2,3,4-tetrahydroisoquinoline, their preparation method and their use as fungicides CYP1A1, CBR3, HAAO ALDH1A1 203/4885KDM4E 1424/4885MAPT 4239/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.