SCHEMBL5751212

SCHEMBL5751212

NNC(=O)Cc1cnc(=O)[nH]c1

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
AOC3 Q16853 14/20 0.42
MET P08581 1/20 0.39
AOC2 O75106 3/20 0.37
KDM6B O15054 1/20 0.37
KDM4A O75164 1/20 0.37
KDM5A P29375 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5988807 0.79 GABRA1 (0.46) CYP3A4MET
SCHEMBL25237063 0.74 NOS2 (0.56) CYP1A2CYP3A4CYP2C9AOC3AOC2
SCHEMBL5988224 0.69 CYP1A2 (0.56) CYP1A2CYP3A4CYP2C9AOC3AOC2
SCHEMBL2827343 0.68 CYP1A2 (0.58) CYP1A2CYP3A4CYP2C9AOC3AOC2
SCHEMBL11796135 0.67 AOC2 (0.66) CYP1A2CYP3A4CYP2C9AOC3AOC2
SCHEMBL29068210 0.66 NPC1 (0.35) CYP1A2CYP3A4MET
SCHEMBL2495046 0.65 MEN1 (0.55) CYP1A2CYP3A4CYP2C9AOC3AOC2
SCHEMBL14424070 0.65 MEN1 (0.38) CYP2C9MET
SCHEMBL968125 0.63 CYP1A2 (0.62) CYP1A2CYP3A4CYP2C9AOC3AOC2
SCHEMBL2222457 0.63 NNMT (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1644362-A2 INDOLINONE HYDRAZIDES AS C-MET INHIBITORS Sugen, Inc. (US) 2006-04-12 EP disclosed
US-20060009493-A1 Indolinone hydrazides as c-Met inhibitors SUGEN, INC. 2006-01-12 US disclosed
WO-2005005378-A2 INDOLINONE HYDRAZIDES AS C-MET INHIBITORS SUGEN, INC. (US) 2005-01-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060009493-A1 Indolinone hydrazides as c-Met inhibitors MET, IGF1R, ROS1 CYP1A2 966/4885CYP3A4 894/4885CYP2C9 792/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.