SCHEMBL5752901

SCHEMBL5752901

Fc1ccc(OC(OC(Oc2ccc(F)cc2)C2CO2)C2CO2)cc1

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.33
PPARG P37231 1/20 0.32
PPARA Q07869 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL726736 0.81 TDP1 (0.41) ALDH1A1
SCHEMBL18920686 0.74 ALDH1A1 (0.37) ALDH1A1
Acrylic Acid SCHEMBL4400635 0.69 THRB (0.35) ALDH1A1PPARGPPARARAB9A
SCHEMBL7227399 0.69 IDO1 (0.38)
SCHEMBL7235653 0.69 IDO1 (0.38)
SCHEMBL6843632 0.69 FUT7 (0.39) PPARGPPARA
SCHEMBL2780633 0.67 ADRA2A (0.43) ALDH1A1RAB9A
SCHEMBL9587807 0.67 TDP1 (0.39)
SCHEMBL11218368 0.66 ACHE (0.45) ALDH1A1
SCHEMBL9488060 0.66

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1099692-B1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES EISAI CO LTD (JP) 2006-05-03 EP disclosed
US-6737425-B1 SUCH AS 1-((4-CYANO-5-METHYL-4-PHENYL)HEXYL)-4-(2-(4-FLUORO -PHENOXY)ETHYL)PIPERAZINE; NERVE SELECTIVE CALCIUM ANTAGONISTS EISAI CO., LTD. (JP) 2004-05-18 US disclosed
CN-1310709-A N, N-substituted cyclic amine derivatives EISAI CO LTD (JP) 2001-08-29 CN disclosed
EP-1099692-A1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES Eisai Co., Ltd. (JP) 2001-05-16 EP disclosed