SCHEMBL5756844

SCHEMBL5756844

CC(=O)Oc1ccc(F)cc1C(C)=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFD P00746 2/20 0.51
KDM4E B2RXH2 7/20 0.50
ALDH1A1 P00352 5/20 0.50
HSD17B10 Q99714 3/20 0.50
TSHR P16473 2/20 0.50
PTGS1 P23219 2/20 0.50
PTGS2 P35354 2/20 0.50
HPGD P15428 2/20 0.50
ESR1 P03372 1/20 0.50
ITGB3 P05106 1/20 0.50
ITGA2B P08514 1/20 0.50
HMGB1 P09429 1/20 0.50
GGT1 P19440 1/20 0.50
BLM P54132 1/20 0.50
NAPRT Q6XQN6 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
HTT P42858 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
KMT2A Q03164 2/20 0.45
LMNA P02545 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1162085 0.87 CFD (0.69) CFDKDM4EALDH1A1HSD17B10TSHR
SCHEMBL1162227 0.86 CFD (0.49) CFDKDM4EALDH1A1HSD17B10TSHR
SCHEMBL43492 0.83 PIN1 (0.49) KDM4EALDH1A1HSD17B10HTTSMN1; SMN2
SCHEMBL28383775 0.83 ALDH1A1 (0.49) CFDKDM4EALDH1A1HSD17B10TSHR
SCHEMBL5755257 0.82 TSHR (0.58) CFDKDM4EALDH1A1HSD17B10TSHR
SCHEMBL5756842 0.82 ALDH1A1 (0.44) ALDH1A1TSHRHTTSMN1; SMN2KMT2A
SCHEMBL823700 0.81 CYP4F2 (0.50) CFDKDM4EALDH1A1HSD17B10TSHR
SCHEMBL22950969 0.79 KDM4E (0.61) CFDKDM4EALDH1A1HSD17B10TSHR
SCHEMBL195552 0.79 KMT2A (0.60) CFDKDM4EALDH1A1HSD17B10TSHR
SCHEMBL789388 0.79 PTGDR2 (0.63) CFDKDM4EALDH1A1HSD17B10TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102015641-B Heterocyclic compound TAKEDA PHARMACEUTICAL 2014-01-01 CN disclosed
CN-102015641-A Heterocyclic compound TAKEDA PHARMACEUTICAL 2011-04-13 CN disclosed
EP-1099692-B1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES EISAI CO LTD (JP) 2006-05-03 EP disclosed
US-6737425-B1 SUCH AS 1-((4-CYANO-5-METHYL-4-PHENYL)HEXYL)-4-(2-(4-FLUORO -PHENOXY)ETHYL)PIPERAZINE; NERVE SELECTIVE CALCIUM ANTAGONISTS EISAI CO., LTD. (JP) 2004-05-18 US disclosed
EP-1099692-A1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES Eisai Co., Ltd. (JP) 2001-05-16 EP disclosed