SCHEMBL5757611

SCHEMBL5757611

CN(C)CC(O)Cn1nc(C2=C(c3cn(C)c4ccccc34)C(=O)NC2=O)c2ccccc21

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 15/20 0.59
CCNE2 O96020 2/20 0.56
CDK4 P11802 2/20 0.56
CCND1 P24385 2/20 0.56
CCNE1 P24864 2/20 0.56
CDK2 P24941 2/20 0.56
PRKCA P17252 9/20 0.56
PRKCG P05129 8/20 0.56
PRKCB P05771 8/20 0.56
PRKCD Q05655 5/20 0.53
PIM1 P11309 1/20 0.52
PRKACA P17612 1/20 0.52
PRKACG P22612 1/20 0.52
PRKACB P22694 1/20 0.52
KCNH2 Q12809 3/20 0.52
PRKCZ Q05513 2/20 0.52
IDH1 O75874 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3777462 0.92 GSK3B (0.53) GSK3BCCNE2CDK4CCND1CCNE1
SCHEMBL5756702 0.87 GSK3B (0.71) GSK3BCCNE2CDK4CCND1CCNE1
SCHEMBL5758314 0.84 CAMK2D (0.62) GSK3BCCNE2CDK4CCND1CCNE1
SCHEMBL3775416 0.82 GSK3B (0.79) GSK3BCCNE2CDK4CCND1CCNE1
SCHEMBL3775971 0.80 GSK3B (0.61) GSK3BCDK4CCND1CDK2PRKCA
SCHEMBL8249349 0.77 CDK2 (0.74) GSK3BCCNE2CDK4CCND1CCNE1
SCHEMBL5755763 0.75 GSK3B (0.64) GSK3BCCNE2CDK4CCND1CCNE1
SCHEMBL5757844 0.75 GSK3B (0.67) GSK3BCDK4CCND1CDK2PRKCA
SCHEMBL30319849 0.74 CCNE2 (1.00) GSK3BCCNE2CDK4CCND1CCNE1
SCHEMBL5686048 0.74 CCNE2 (1.00) GSK3BCCNE2CDK4CCND1CCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1362047-B1 INDAZOLYL-SUBSTITUTED PYRROLINE COMPOUNDS AS KINASE INHIBITORS ORTHO MCNEIL PHARM INC (US) 2006-05-17 EP disclosed