SCHEMBL5757744

SCHEMBL5757744

O=C(O)c1cnc2cc(-c3cccs3)ccc2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGAM O43451 1/20 0.54
SRPK1 Q96SB4 1/20 0.53
RPS6KB2 Q9UBS0 1/20 0.53
EGLN1 Q9GZT9 1/20 0.50
HDAC2 Q92769 4/20 0.49
PDGFRB P09619 1/20 0.44
PDGFRA P16234 1/20 0.44
CHEK1 O14757 1/20 0.43
CHEK2 O96017 1/20 0.43
KDM4E B2RXH2 3/20 0.43
MAPT P10636 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
CYP1A2 P05177 1/20 0.42
HPGD P15428 1/20 0.42
CYP2C19 P33261 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
HDAC3 O15379 3/20 0.41
HDAC1 Q13547 3/20 0.41
HPGDS O60760 1/20 0.41
PGR P06401 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL528875 0.89 MGAM (0.54) MGAMSRPK1RPS6KB2EGLN1HDAC2
SCHEMBL5757063 0.82 MAOB (0.53) HDAC2PDGFRBPDGFRAKDM4EMAPT
SCHEMBL28055368 0.78 MGAM (0.60) MGAMPDGFRBPDGFRAKDM4EHPGDS
SCHEMBL5762283 0.77 PDGFRB (0.45) RPS6KB2HDAC2PDGFRBPDGFRACHEK1
SCHEMBL10080493 0.76 SRPK1 (0.57) SRPK1RPS6KB2EGLN1HDAC2KDM4E
SCHEMBL69368 0.74 MGAM (0.68) MGAMPDGFRBPDGFRAKDM4EMAPT
SCHEMBL27402367 0.74 PDGFRB (0.58) RPS6KB2PDGFRBPDGFRAKDM4EMAPT
SCHEMBL5762231 0.74 PDGFRB (0.45) RPS6KB2HDAC2PDGFRBPDGFRAKDM4E
SCHEMBL569420 0.74 CYP2E1 (0.50) SRPK1RPS6KB2EGLN1HDAC2CHEK1
SCHEMBL420705 0.72 KDM4E (0.55) SRPK1RPS6KB2EGLN1HDAC2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1270571-B1 Heterocyclic compounds, their production and use TAKEDA PHARMACEUTICAL (JP) 2006-09-06 EP disclosed
EP-1270571-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-01-02 EP disclosed
US-6211215-B1 AROMATIC HETEROCYCLIC COMPOUND WITH AZOLE COMPOUND TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-04-03 US disclosed
EP-0912562-A1 HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1999-05-06 EP disclosed
WO-1998003505-A2 HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-01-29 WO disclosed