SCHEMBL5757978

SCHEMBL5757978

OCc1ncc(-c2cccs2)s1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.51
SLC5A2 P31639 6/20 0.44
ALDH1A1 P00352 5/20 0.41
GAA P10253 4/20 0.41
MAPT P10636 3/20 0.41
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
HTT P42858 1/20 0.41
LTA4H P09960 1/20 0.41
CYP2E1 P05181 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2A6 P11509 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2B6 P20813 1/20 0.39
FYN P06241 1/20 0.39
KDM4E B2RXH2 3/20 0.39
L3MBTL1 Q9Y468 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19721706 0.76 KDM4E (0.46) DPP4ALDH1A1GAAMAPTNPC1
SCHEMBL2226003 0.76 ERCC5 (0.63) SLC5A2CYP3A4CYP2C9ERCC5FEN1
SCHEMBL18876350 0.75 MEN1 (0.41) DPP4ALDH1A1GAAMAPTNPC1
SCHEMBL3072249 0.75 KDM4E (0.48) DPP4ALDH1A1GAAMAPTNPC1
SCHEMBL19501428 0.74 ALDH1A1 (0.41) DPP4ALDH1A1GAAMAPTNPC1
SCHEMBL956185 0.73 ALDH1A1 (0.52) ALDH1A1GAAMAPTNPC1RAB9A
SCHEMBL3232148 0.73 CES1 (0.50) ALDH1A1GAAMAPTNPC1RAB9A
SCHEMBL869424 0.72 KDM4E (0.50) ALDH1A1GAAMAPTNPC1RAB9A
SCHEMBL8178162 0.71 CYP11B1 (0.56) DPP4ALDH1A1GAAMAPTNPC1
SCHEMBL5759550 0.71 DPP4 (0.53) DPP4SLC5A2ALDH1A1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1270571-B1 Heterocyclic compounds, their production and use TAKEDA PHARMACEUTICAL (JP) 2006-09-06 EP disclosed
EP-1270571-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-01-02 EP disclosed
CN-1349990-A Heterocyclic compound, its preparation and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-05-22 CN disclosed
CN-1077107-C Heterocyclic compounds, their preparation and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-01-02 CN disclosed
US-6211215-B1 AROMATIC HETEROCYCLIC COMPOUND WITH AZOLE COMPOUND TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-04-03 US disclosed
CN-1223653-A Heterocyclic compounds, their preparation and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1999-07-21 CN disclosed
EP-0912562-A1 HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1999-05-06 EP disclosed
WO-1998003505-A2 HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-01-29 WO disclosed