SCHEMBL5758945

SCHEMBL5758945

O=C(c1ccccc1)C1CCN(CCCN(C(=O)Cc2ccc(Cl)c(Cl)c2)c2ccccc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.54
CCR5 P51681 9/20 0.49
HTR2A P28223 1/20 0.48
SIGMAR1 Q99720 2/20 0.46
S1PR5 Q9H228 1/20 0.46
CHRM2 P08172 1/20 0.45
CHRM3 P20309 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5758374 0.86 CCR5 (0.60) CCR5
SCHEMBL5758222 0.85 OPRM1 (0.53) SIGMAR1
SCHEMBL5754844 0.81 KCNH2 (0.60) KCNH2CCR5HTR2A
SCHEMBL28602611 0.76 KCNH2 (0.64) KCNH2CCR5SIGMAR1
SCHEMBL6008659 0.73 KCNH2 (0.53) KCNH2CCR5HTR2ASIGMAR1S1PR5
SCHEMBL658329 0.72 HDAC3 (0.49)
SCHEMBL5758044 0.72 KCNH2 (0.62) KCNH2HTR2A
SCHEMBL6009253 0.71 KCNH2 (0.55) KCNH2HTR2ASIGMAR1S1PR5CHRM2
SCHEMBL9647537 0.71 HTR2A (0.72) KCNH2HTR2ASIGMAR1
SCHEMBL8313722 0.71 KCNH2 (0.71) KCNH2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1401821-A4 NOVEL PHENYLALKYL DIAMINE AND AMIDE ANALOGS SK CORP (KR) 2006-05-31 EP claimed
EP-1401821-A1 NOVEL PHENYLALKYL DIAMINE AND AMIDE ANALOGS SK Corporation (KR) 2004-03-31 EP claimed
WO-2002100848-A1 NOVEL PHENYLALKYL DIAMINE AND AMIDE ANALOGS SK CORPORATION (KR) 2002-12-19 WO claimed