SCHEMBL5766533

SCHEMBL5766533

Cc1cccc(Cc2ccc3nnc(-c4ccccc4)n3c2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
KMT2A Q03164 1/20 0.45
KDM4E B2RXH2 2/20 0.44
HSD17B10 Q99714 1/20 0.44
DPP4 P27487 1/20 0.43
NT5E P21589 6/20 0.43
MAPT P10636 2/20 0.42
TP53 P04637 1/20 0.42
NR1H4 Q96RI1 1/20 0.42
MET P08581 2/20 0.41
MAPK14 Q16539 1/20 0.41
LMNA P02545 3/20 0.40
ALDH1A1 P00352 2/20 0.40
PKM P14618 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5763347 0.83 HSD11B1 (0.41) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5766810 0.79 MAPK14 (0.54) MAPK14
SCHEMBL9844320 0.75 KDM4E (0.49) KMT2AKDM4EHSD17B10NT5ETP53
SCHEMBL27681631 0.73 LTA4H (0.55) MEN1CYP3A4KMT2AMAPTTP53
SCHEMBL8085716 0.73 CALM1 (0.55) MEN1KMT2ATP53LMNAL3MBTL1
SCHEMBL5767929 0.72 KDM4E (0.42) KDM4EHSD17B10DPP4NT5EMAPK14
SCHEMBL5772734 0.72 MAPK14 (0.72) MAPK14
SCHEMBL32665199 0.72 KDM4E (0.50) MEN1KMT2AKDM4EHSD17B10DPP4
SCHEMBL6221061 0.71 MLLT1 (0.40) ALDH1A1LTA4H
SCHEMBL23547235 0.71 PIM1 (0.58) KMT2AKDM4EHSD17B10NT5EMET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7321040-B2 Triazolo-pyridines as anti-inflammatory compounds PFIZER INC. (US) 2008-01-22 US disclosed
US-7321040-B2 Triazolo-pyridines as anti-inflammatory compounds PFIZER INC. (US) 2008-01-22 US disclosed
EP-1601672-B1 TRIAZOLO-PYRIDINES AS ANTI-INFLAMMATORY COMPOUNDS PFIZER PROD INC (US) 2006-07-26 EP disclosed