SCHEMBL5769285

SCHEMBL5769285

O=Cc1cn(-c2ccccc2Cl)c2ccccc12

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 13/20 0.56
KDM4E B2RXH2 2/20 0.56
IMPDH2 P12268 1/20 0.51
SMN1; SMN2 Q16637 7/20 0.49
HTT P42858 5/20 0.49
KMT2A Q03164 2/20 0.49
MEN1 O00255 1/20 0.49
LMNA P02545 4/20 0.45
UBE2N P61088 1/20 0.41
MAPT P10636 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
RORC P51449 1/20 0.40
ATM Q13315 1/20 0.40
NPC1 O15118 1/20 0.40
HPGD P15428 1/20 0.40
RAB9A P51151 1/20 0.40
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12627927 0.81 ALDH1A1 (0.56) ALDH1A1KDM4EIMPDH2SMN1; SMN2HTT
SCHEMBL27996103 0.77 ALDH1A1 (0.74) ALDH1A1KDM4EIMPDH2SMN1; SMN2HTT
SCHEMBL4697569 0.77 ALDH1A1 (0.52) ALDH1A1KDM4EIMPDH2SMN1; SMN2HTT
SCHEMBL9412272 0.76 ALDH1A1 (0.78) ALDH1A1KDM4EIMPDH2SMN1; SMN2HTT
SCHEMBL31116748 0.75 RORC (0.42) ALDH1A1KDM4EKMT2AMEN1MAPT
SCHEMBL674179 0.74 ALDH1A1 (0.58) ALDH1A1KDM4EIMPDH2SMN1; SMN2HTT
SCHEMBL5102370 0.74 ALDH1A1 (0.56) ALDH1A1KDM4EIMPDH2SMN1; SMN2HTT
SCHEMBL6869652 0.73 ALDH1A1 (0.53) ALDH1A1KDM4EIMPDH2SMN1; SMN2HTT
SCHEMBL27716107 0.72 RORC (0.52) ALDH1A1SMN1; SMN2KMT2ALMNARORC
SCHEMBL7202295 0.72 ALDH1A1 (0.61) ALDH1A1KDM4EIMPDH2SMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1663202-A1 SUBSTITUTED INDOLES AS INHIBITORS OF POLY (ADP-RIBOSE) POLYMERASE (PARP) Aventis Pharmaceuticals, Inc. (US) 2006-06-07 EP disclosed
WO-2005023246-A1 SUBSTITUTED INDOLES AS INHIBITORS OF POLY (ADP-RIBOSE) POLYMERASE (PARP) AVENTIS PHARMACEUTICALS INC. (US) 2005-03-17 WO disclosed