SCHEMBL5771393

SCHEMBL5771393

Brc1cccc2c1Sc1ccccc1S2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.43
BCHE P06276 4/20 0.36
MAOA P21397 2/20 0.36
SLC6A3 Q01959 2/20 0.36
MEN1 O00255 1/20 0.36
CYP1A2 P05177 1/20 0.36
POLB P06746 1/20 0.36
CYP3A4 P08684 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
ALOX15 P16050 1/20 0.36
ALOX12 P18054 1/20 0.36
CNR1 P21554 1/20 0.36
ACHE P22303 1/20 0.36
PTGS1 P23219 1/20 0.36
SLC6A2 P23975 1/20 0.36
HTR2C P28335 1/20 0.36
PTGS2 P35354 1/20 0.36
SNCA P37840 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30788160 1.00 ALOX5 (0.43) ALOX5BCHEMAOASLC6A3MEN1
SCHEMBL18489034 0.93 ALOX5 (0.34) ALOX5ALDH1A1HDAC6HDAC4HDAC1
SCHEMBL1144919 0.90 MAOA (0.33) ALOX5BCHEMAOASLC6A3MEN1
SCHEMBL10980556 0.84 ALOX5 (0.37) ALOX5BCHESLC6A3SNCA
SCHEMBL18034391 0.83 ALOX5 (0.54) ALOX5BCHEMAOASLC6A3MEN1
SCHEMBL3163268 0.81 MEN1 (0.39) ALOX5MEN1CYP3A4MAPTALOX15
SCHEMBL16545942 0.81 ALOX5 (0.35) ALOX5
SCHEMBL3160482 0.79 ALOX5 (0.39) ALOX5ALOX15TDP1ALDH1A1HPGD
SCHEMBL3185489 0.77 ALOX5 (0.37) ALOX5BCHEMAOASLC6A3MEN1
SCHEMBL2762768 0.76 RECQL (0.39) ALOX5BCHESLC6A3MEN1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 27 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024257964-A1 COMPOUND USED AS ELECTRON BLOCKING LAYER FOR TADF AND ORGANIC LIGHT-EMITTING DEVICE COMPRISING SAME 비피시 주식회사 2024-12-19 WO disclosed
CN-118922416-A Compound and organic light emitting device comprising the same 株式会社LG化学 2024-11-08 CN disclosed
WO-2024101948-A1 COMPOUND AND ORGANIC LIGHT-EMITTING ELEMENT COMPRISING SAME 주식회사 엘지화학 2024-05-16 WO disclosed
WO-2021120838-A1 ORGANIC COMPOUND, ELECTRONIC DEVICE, AND ELECTRONIC APPARATUS 陕西莱特光电材料股份有限公司 2021-06-24 WO disclosed
US-11008280-B2 Compound for organic electric element, organic electric element using same, and electronic device comprising same organic electronic element DUK SAN NEOLUX CO., LTD. (KR) 2021-05-18 US disclosed
EP-3326998-B1 COMPOUND FOR ORGANIC ELECTRIC ELEMENT, ORGANIC ELECTRIC ELEMENT COMPRISING THE SAME, AND ELECTRONIC DEVICE THEREOF DUK SAN NEOLUX CO LTD (KR) 2020-12-02 EP disclosed
EP-3326998-B1 COMPOUND FOR ORGANIC ELECTRIC ELEMENT, ORGANIC ELECTRIC ELEMENT COMPRISING THE SAME, AND ELECTRONIC DEVICE THEREOF DUK SAN NEOLUX CO LTD (KR) 2020-12-02 EP disclosed
US-10797247-B2 Compound for organic electric element, organic electric element comprising the same and electronic device thereof DUK SAN NEOLUX CO., LTD. (KR) 2020-10-06 US disclosed
CN-107922311-B Compound for organic electric element, organic electric element using same, and electronic device using same 德山新勒克斯有限公司 2019-12-17 CN disclosed
US-10468606-B2 Compound for organic electric element, organic electric element comprising the same, and electronic device thereof DUK SAN NEOLUX CO., LTD. (KR) 2019-11-05 US disclosed
WO-2017188676-A1 COMPOUND FOR ORGANIC ELECTRONIC ELEMENT, ORGANIC ELECTRONIC ELEMENT USING SAME, AND ELECTRONIC DEVICE THEREOF 덕산네오룩스 주식회사 2017-11-02 WO disclosed
WO-2017188676-A1 COMPOUND FOR ORGANIC ELECTRONIC ELEMENT, ORGANIC ELECTRONIC ELEMENT USING SAME, AND ELECTRONIC DEVICE THEREOF 덕산네오룩스 주식회사 2017-11-02 WO disclosed
WO-2017188655-A1 COMPOUND FOR ORGANIC ELECTRIC ELEMENT, ORGANIC ELECTRIC ELEMENT USING SAME, AND ELECTRONIC DEVICE COMPRISING SAME ORGANIC ELECTRONIC ELEMENT 덕산네오룩스 주식회사 2017-11-02 WO disclosed
WO-2017119654-A1 COMPOUND FOR ORGANIC ELECTRONIC ELEMENT, ORGANIC ELECTRONIC ELEMENT USING SAME AND ELECTRONIC APPARATUS THEREFOR 덕산네오룩스 주식회사 2017-07-13 WO disclosed
US-20160035983-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE IN ELECTRO-OPTICAL OR OPTO-ELECTRONIC DEVICES POWER OLEDS LTD (GB) 2016-02-04 US disclosed
US-20160035983-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE IN ELECTRO-OPTICAL OR OPTO-ELECTRONIC DEVICES POWER OLEDS LTD (GB) 2016-02-04 US disclosed
WO-2014167286-A2 HETEROCYCLIC COMPOUNDS AND THEIR USE IN ELECTRO-OPTICAL OR OPTO-ELECTRONIC DEVICES POWER OLEDS LIMITED (GB) 2014-10-16 WO disclosed
EP-1654257-A1 AMINOPYRONES AND THEIR USE AS ATM INHIBITORS Kudos Pharmaceuticals Limited (GB) 2006-05-10 EP disclosed
WO-2005016919-A1 AMINOPYRONES AND THEIR USE AS ATM INHIBITORS KUDOS PHARMACEUTICALS LIMITED (GB) 2005-02-24 WO disclosed
US-5095157-A Friedel-crafts catalyst BAYER AKTIENGESELLSCHAFT (DE) 1992-03-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10797247-B2 Compound for organic electric element, organic electric element comprising the same and electronic device thereof PIEZO1, ORAI2, TRPV2 ALOX5 2015/4885BCHE 3051/4885MAOA 2924/4885
US-10468606-B2 Compound for organic electric element, organic electric element comprising the same, and electronic device thereof PIEZO1, OCIAD1, OR10J3 ALOX5 1235/4885BCHE 1835/4885MAOA 779/4885
US-20160035983-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE IN ELECTRO-OPTICAL OR OPTO-ELECTRONIC DEVICES NAT1, SLCO2A1, SLCO2B1 ALOX5 445/4885BCHE 2982/4885MAOA 407/4885
US-11008280-B2 Compound for organic electric element, organic electric element using same, and electronic device comprising same organic electronic element ORAI2, PIEZO1, ORC3 ALOX5 1003/4885BCHE 1252/4885MAOA 1922/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.