SCHEMBL5773732

SCHEMBL5773732

CC(C)S(=O)(=O)n1c(NCc2cccnc2)nc2ccc(C=N)cc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.38
ALDH1A1 P00352 3/20 0.38
GAA P10253 2/20 0.38
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 2/20 0.38
CYP2D6 P10635 2/20 0.38
CYP2C19 P33261 2/20 0.38
CYP2C9 P11712 1/20 0.38
GSK3B P49841 3/20 0.38
PDE9A O76083 1/20 0.38
MAPK14 Q16539 1/20 0.37
RAB9A P51151 2/20 0.37
CD274 Q9NZQ7 1/20 0.37
MAPK1 P28482 2/20 0.37
KMT2A Q03164 2/20 0.37
POLB P06746 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
HSD17B10 Q99714 2/20 0.36
USP2 O75604 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5774512 0.88 ALDH1A1 (0.40) KDM4EALDH1A1GAACYP2C19MAPK14
SCHEMBL5773725 0.85 MAPK14 (0.42) KDM4EALDH1A1GAACYP1A2CYP3A4
SCHEMBL5773723 0.83 MAPK14 (0.41) KDM4EALDH1A1GAACYP1A2CYP3A4
SCHEMBL5770367 0.80 MAPK14 (0.41) GAACYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL5770827 0.80 TP53 (0.48) ALDH1A1GAACYP1A2CYP3A4CYP2D6
SCHEMBL5767550 0.77 MAPK14 (0.38) CYP3A4MAPK14
SCHEMBL5769574 0.77 PI4KB (0.36) CYP3A4MAPK14
SCHEMBL18058953 0.74 THRB (0.50) KDM4EALDH1A1GAACYP1A2CYP3A4
SCHEMBL5772161 0.74 PI4KB (0.39) KDM4EALDH1A1CYP3A4CYP2C19CYP2C9
SCHEMBL18057139 0.74 MAPK14 (0.44) ALDH1A1GAACYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1554272-B1 BENZIMIDAZOLES AND BENZOTHIAZOLES AS INHIBITORS OF MAP KINASE LILLY CO ELI (US) 2006-10-25 EP disclosed