SCHEMBL5776715

SCHEMBL5776715

Clc1cccc2nc(C3[CH]NCCC3)ccc12

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
CYP1A2 P05177 1/20 0.32
CLK4 Q9HAZ1 1/20 0.32
ACP1 P24666 1/20 0.32
GUSB P08236 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5776458 0.79 CYP3A4 (0.41) CYP1A2
SCHEMBL4155227 0.64 SLC18A3 (0.42) CYP1A2
SCHEMBL239860 0.63 CYP1A2 (0.46) PDE3BPDE3ACYP1A2GUSB
SCHEMBL29746469 0.63 CYP1A2 (0.46) PDE3BPDE3ACYP1A2GUSB
SCHEMBL5779423 0.63 CYP1A2 (0.40) CYP1A2
SCHEMBL5779681 0.62 IRAK4 (0.36)
SCHEMBL8889348 0.61 MEN1 (0.50) CYP1A2
SCHEMBL3071480 0.60 BACE1 (0.60) CYP1A2
SCHEMBL29980068 0.60 CYP1A2 (0.42) PDE3BPDE3ACYP1A2GUSB
SCHEMBL2757268 0.60 ALDH1A1 (0.51) PDE3BPDE3ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633735-A1 DERIVATIVES OF PIPERIDINYL- AND PIPERAZINYL-ALKYL CARBAMATES, PREPARATION METHODS THEREOF AND APPLICATION OF SAME IN THERAPEUTICS Sanofi-Aventis (FR) 2006-03-15 EP disclosed
WO-2004099176-A1 DERIVATIVES OF PIPERIDINYL- AND PIPERAZINYL-ALKYL CARBAMATES, PREPARATION METHODS THEREOF AND APPLICATION OF SAME IN THERAPEUTICS SANOFI-AVENTIS (FR) 2004-11-18 WO disclosed