SCHEMBL5778370

SCHEMBL5778370

CC(Cc1ccc2ncccc2c1)S(C)(=O)=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.48
ALDH1A1 P00352 3/20 0.45
NPC1 O15118 3/20 0.44
POLB P06746 2/20 0.44
RAB9A P51151 1/20 0.44
DAO P14920 1/20 0.43
CHKA P35790 1/20 0.42
MAPT P10636 2/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
PDE10A Q9Y233 2/20 0.42
FCER2 P06734 1/20 0.42
MET P08581 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
HDAC3 O15379 1/20 0.41
KDM4E B2RXH2 1/20 0.41
TP53 P04637 1/20 0.41
HSP90AA1 P07900 1/20 0.41
HSP90AB1 P08238 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL113636 0.82 ALDH1A1 (0.53) ACACBALDH1A1NPC1POLBRAB9A
SCHEMBL29873370 0.82 ALDH1A1 (0.53) ACACBALDH1A1NPC1POLBRAB9A
SCHEMBL26854390 0.79 ALDH1A1 (0.50) ACACBALDH1A1NPC1POLBRAB9A
SCHEMBL5778919 0.77 GLO1 (0.37) ALDH1A1MAPTMEN1KMT2AKDM4E
SCHEMBL28308974 0.76 ACACB (0.45) ACACBALDH1A1NPC1POLBRAB9A
SCHEMBL934232 0.76 FCER2 (0.53) ACACBALDH1A1NPC1POLBRAB9A
SCHEMBL4049830 0.75 ALDH1A1 (0.46) ALDH1A1NPC1POLBRAB9ADAO
SCHEMBL27620527 0.75 NPC1 (0.52) ACACBALDH1A1NPC1POLBRAB9A
SCHEMBL2297609 0.74 PKM (0.55) ACACBALDH1A1NPC1POLBMAPT
SCHEMBL5783367 0.74 PKM (0.55) ACACBALDH1A1NPC1POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1635829-A1 8-(3-BIARYL)PHENYLQUINOLINE PHOSPHODIESTERASE-4-INHIBITORS Merck Frosst Canada Ltd. (CA) 2006-03-22 EP claimed
WO-2004096220-A1 8-(3-BIARYL)PHENYLQUINOLINE PHOSPHODIESTERASE-4-INHIBITORS MERCK FROSST CANADA LTD. (CA) 2004-11-11 WO claimed