SCHEMBL5780422

SCHEMBL5780422

C=CC[C@H]1N(C(=O)c2cccc(F)c2F)c2ccc(F)cc2C12CCNCC2

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.36
HPGD P15428 1/20 0.34
GNRHR P30968 2/20 0.33
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32
KCNH2 Q12809 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32
DPP4 P27487 1/20 0.31
ATM Q13315 1/20 0.31
PSEN1 P49768 2/20 0.31
PSEN2 P49810 2/20 0.31
APH1B Q8WW43 2/20 0.31
NCSTN Q92542 2/20 0.31
APH1A Q96BI3 2/20 0.31
PSENEN Q9NZ42 2/20 0.31
DRD2 P14416 1/20 0.31
USP2 O75604 2/20 0.31
CYP2D6 P10635 2/20 0.31
GRM5 P41594 1/20 0.31
ALOX15 P16050 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5599667 0.90 ATM (0.37) HPGDHCRTR1HCRTR2ATMDRD2
SCHEMBL5786885 0.89 GNRHR (0.33) GNRHRKCNH2PTGDR2DPP4PSEN1
SCHEMBL5786887 0.87 GNRHR (0.41) P2RX7GNRHRKCNH2PSEN1PSEN2
SCHEMBL5600002 0.86 P2RX7 (0.37) P2RX7HPGDGNRHRHCRTR1HCRTR2
SCHEMBL5599502 0.85 GNRHR (0.32) GNRHRKCNH2DPP4
SCHEMBL5778222 0.84 SMYD3 (0.34) GNRHRKCNH2ALDH1A1
SCHEMBL5600190 0.84 GNRHR (0.36) P2RX7GNRHRKCNH2PSEN1PSEN2
SCHEMBL5599977 0.83 GNRHR (0.34) GNRHRKCNH2DPP4PSEN1PSEN2
SCHEMBL5788610 0.83 GNRHR (0.34) GNRHRKCNH2DPP4PSEN1PSEN2
SCHEMBL5599482 0.83 HTT (0.37) ALDH1A1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1716148-A2 NOVEL SPIROINDOLINE OR SPIROISOQUINOLINE COMPOUNDS, METHODS OF USE AND COMPOSITIONS THEREOF Arena Pharmaceuticals, Inc. (US) 2006-11-02 EP claimed
WO-2005063745-A2 NOVEL SPIROINDOLINE OR SPIROISOQUINOLINE COMPOUNDS, METHODS OF USE AND COMPOSITIONS THEREOF ARENA PHARMACEUTICALS, INC. (US) 2005-07-14 WO claimed